日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of New KCNT1-Epilepsy Drugs by In Silico, Cell, and Drosophila Modeling

利用计算机模拟、细胞和果蝇模型鉴定新的KCNT1癫痫药物

Ricos, Michael G; Cole, Bethan A; Hussain, Rashid; Rychkov, Grigori Y; Shaukat, Zeeshan; Pilati, Nadia; Muench, Stephen P; Simmons, Katie J; Dibbens, Leanne M; Lippiat, Jonathan D

Targeting Ca(2+) Signaling in the Initiation, Promotion and Progression of Hepatocellular Carcinoma

靶向Ca(2+)信号通路在肝细胞癌的发生、发展和进展中的作用

Ali, Eunus S; Rychkov, Grigori Y; Barritt, Greg J

Cyclic analogues of α-conotoxin Vc1.1 inhibit colonic nociceptors and provide analgesia in a mouse model of chronic abdominal pain

α-芋螺毒素Vc1.1的环状类似物可抑制结肠伤害感受器,并在慢性腹痛小鼠模型中发挥镇痛作用

Castro, Joel; Grundy, Luke; Deiteren, Annemie; Harrington, Andrea M; O'Donnell, Tracey; Maddern, Jessica; Moore, Jessi; Garcia-Caraballo, Sonia; Rychkov, Grigori Y; Yu, Rilei; Kaas, Quentin; Craik, David J; Adams, David J; Brierley, Stuart M

NaV1.1 inhibition can reduce visceral hypersensitivity

NaV1.1抑制可降低内脏高敏感性

Salvatierra, Juan; Castro, Joel; Erickson, Andelain; Li, Qian; Braz, Joao; Gilchrist, John; Grundy, Luke; Rychkov, Grigori Y; Deiteren, Annemie; Rais, Rana; King, Glenn F; Slusher, Barbara S; Basbaum, Allan; Pasricha, Pankaj J; Brierley, Stuart M; Bosmans, Frank

Chronic linaclotide treatment reduces colitis-induced neuroplasticity and reverses persistent bladder dysfunction

长期使用利那洛肽治疗可减少结肠炎引起的神经可塑性并逆转持续性膀胱功能障碍

Grundy, Luke; Harrington, Andrea M; Castro, Joel; Garcia-Caraballo, Sonia; Deiteren, Annemie; Maddern, Jessica; Rychkov, Grigori Y; Ge, Pei; Peters, Stefanie; Feil, Robert; Miller, Paul; Ghetti, Andre; Hannig, Gerhard; Kurtz, Caroline B; Silos-Santiago, Inmaculada; Brierley, Stuart M

Multiple sodium channel isoforms mediate the pathological effects of Pacific ciguatoxin-1

多种钠通道亚型介导太平洋雪卡毒素-1的病理效应

Inserra, Marco C; Israel, Mathilde R; Caldwell, Ashlee; Castro, Joel; Deuis, Jennifer R; Harrington, Andrea M; Keramidas, Angelo; Garcia-Caraballo, Sonia; Maddern, Jessica; Erickson, Andelain; Grundy, Luke; Rychkov, Grigori Y; Zimmermann, Katharina; Lewis, Richard J; Brierley, Stuart M; Vetter, Irina

Selective spider toxins reveal a role for the Nav1.1 channel in mechanical pain

选择性蜘蛛毒素揭示了Nav1.1通道在机械性疼痛中的作用

Osteen, Jeremiah D; Herzig, Volker; Gilchrist, John; Emrick, Joshua J; Zhang, Chuchu; Wang, Xidao; Castro, Joel; Garcia-Caraballo, Sonia; Grundy, Luke; Rychkov, Grigori Y; Weyer, Andy D; Dekan, Zoltan; Undheim, Eivind A B; Alewood, Paul; Stucky, Cheryl L; Brierley, Stuart M; Basbaum, Allan I; Bosmans, Frank; King, Glenn F; Julius, David

Respiratory distress and perinatal lethality in Nedd4-2-deficient mice.

Nedd4-2 缺陷小鼠出现呼吸窘迫和围产期死亡

Boase Natasha A, Rychkov Grigori Y, Townley Scott L, Dinudom Anuwat, Candi Eleanora, Voss Anne K, Tsoutsman Tatiana, Semsarian Chris, Melino Gerry, Koentgen Frank, Cook David I, Kumar Sharad

Functional complementation of truncated human skeletal-muscle chloride channel (hClC-1) using carboxyl tail fragments

利用羧基尾片段对截短的人类骨骼肌氯离子通道(hClC-1)进行功能互补

Wu, Weiping; Rychkov, Grigori Y; Hughes, Bernard P; Bretag, Allan H

Arachidonic acid inhibits the store-operated Ca2+ current in rat liver cells

花生四烯酸抑制大鼠肝细胞中由储存操纵的Ca2+电流。

Rychkov, Grigori Y; Litjens, Tom; Roberts, Michael L; Barritt, Greg J