日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Characterization of the second conserved domain in the heme uptake protein HtaA from Corynebacterium diphtheriae

白喉棒状杆菌血红素摄取蛋白HtaA第二个保守结构域的特征分析

Uluisik, Rizvan C; Akbas, Neval; Lukat-Rodgers, Gudrun S; Adrian, Seth A; Allen, Courtni E; Schmitt, Michael P; Rodgers, Kenton R; Dixon, Dabney W

An Ultra-High-Throughput Screen for Catalytic Inhibitors of Serine/Threonine Protein Phosphatases Types 1 and 5 (PP1C and PP5C)

丝氨酸/苏氨酸蛋白磷酸酶1型和5型(PP1C和PP5C)催化抑制剂的超高通量筛选

Swingle, Mark; Volmar, Claude-Henry; Saldanha, S Adrian; Chase, Peter; Eberhart, Christina; Salter, Edward A; D'Arcy, Brandon; Schroeder, Chad E; Golden, Jennifer E; Wierzbicki, Andrzej; Hodder, Peter; Honkanen, Richard E

Gold nanoparticles grown inside carbon nanotubes: synthesis and electrical transport measurements

碳纳米管内生长的金纳米粒子:合成及电输运测量

Segura, Rodrigo A; Contreras, Claudia; Henriquez, Ricardo; Häberle, Patricio; Acuña, José Javier S; Adrian, Alvaro; Alvarez, Pedro; Hevia, Samuel A

Implementing fluorescence anisotropy screening and crystallographic analysis to define PKA isoform-selective activation by cAMP analogs

运用荧光各向异性筛选和晶体学分析来确定cAMP类似物对PKA亚型的选择性激活作用

Brown, Simon H J; Cheng, Cecilia Y; Saldanha, S Adrian; Wu, Jian; Cottam, Howard B; Sankaran, Banumathi; Taylor, Susan S

Design, synthesis and SAR analysis of novel potent and selective small molecule antagonists of NPBWR1 (GPR7)

NPBWR1 (GPR7) 新型高效选择性小分子拮抗剂的设计、合成及构效关系分析

Urbano, Mariangela; Guerrero, Miguel; Zhao, Jian; Velaparthi, Subash; Saldanha, S Adrian; Chase, Peter; Wang, Zhiwei; Civelli, Olivier; Hodder, Peter; Schaeffer, Marie-Therese; Brown, Steven; Rosen, Hugh; Roberts, Edward

Small-molecule proteostasis regulators for protein conformational diseases

用于蛋白质构象疾病的小分子蛋白质稳态调节剂

Calamini, Barbara; Silva, Maria Catarina; Madoux, Franck; Hutt, Darren M; Khanna, Shilpi; Chalfant, Monica A; Saldanha, S Adrian; Hodder, Peter; Tait, Bradley D; Garza, Dan; Balch, William E; Morimoto, Richard I

Selective and brain penetrant neuropeptide y y2 receptor antagonists discovered by whole-cell high-throughput screening

通过全细胞高通量筛选发现选择性和脑渗透性神经肽 y y2 受体拮抗剂

Shaun P Brothers, S Adrian Saldanha, Timothy P Spicer, Michael Cameron, Becky A Mercer, Peter Chase, Patricia McDonald, Claes Wahlestedt, Peter S Hodder

Small molecule activators of TRPML3

TRPML3的小分子激活剂

Grimm, Christian; Jörs, Simone; Saldanha, S Adrian; Obukhov, Alexander G; Pan, Bifeng; Oshima, Kazuo; Cuajungco, Math P; Chase, Peter; Hodder, Peter; Heller, Stefan

Virtual ligand screening of the p300/CBP histone acetyltransferase: identification of a selective small molecule inhibitor

p300/CBP 组蛋白乙酰转移酶的虚拟配体筛选:选择性小分子抑制剂的鉴定

Erin M Bowers, Gai Yan, Chandrani Mukherjee, Andrew Orry, Ling Wang, Marc A Holbert, Nicholas T Crump, Catherine A Hazzalin, Glen Liszczak, Hua Yuan, Cecilia Larocca, S Adrian Saldanha, Ruben Abagyan, Yan Sun, David J Meyers, Ronen Marmorstein, Louis C Mahadevan, Rhoda M Alani, Philip A Cole

High throughput screening of potentially selective MMP-13 exosite inhibitors utilizing a triple-helical FRET substrate

利用三螺旋 FRET 底物高通量筛选潜在选择性 MMP-13 外部抑制剂

Janelle L Lauer-Fields, Dmitriy Minond, Peter S Chase, Pierre E Baillargeon, S Adrian Saldanha, Roma Stawikowska, Peter Hodder, Gregg B Fields