Tissue distribution and retention drives efficacy of rapidly clearing VHL-based PROTACs
组织分布和保留决定了快速清除基于 VHL 的 PROTAC 的功效
期刊:Commun Med (Lond)
影响因子:
doi:10.1038/s43856-024-00505-y
Donglu Zhang, Bin Ma, Peter S Dragovich, Li Ma, Shu Chen, Eugene C Chen, Xiaofen Ye, Joyce Liu, Jennifer Pizzano, Elizabeth Bortolon, Emily Chan, Xing Zhang, Yi-Chen Chen, Elizabeth S Levy, Robert L Yauch, S Cyrus Khojasteh, Cornelis E C A Hop