日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Integrative Multi-Omics Analysis Identifies Nuclear Factor I as a Key Driver of Dysregulated Purine Metabolism in DIPG

整合多组学分析揭示核因子I是DIPG中嘌呤代谢紊乱的关键驱动因素

Mersich, Ian; Congrove, Sunny; Horchar, Matthew; Caceres, Roman; Muraleedharan, Ranjithmenon; Desai, Janki; Desai, Pankaj; Sallans, Larry; Reisz, Julie A; Grier, Abby; Hass, Matthew R; Donmez, Omer; Yin, Cailing; Weirauch, Matthew T; Kottyan, Leah; Stevenson, Charles B; Sun, Claire; de Blank, Peter; Pillay-Smiley, Natasha; Hummel, Trent R; Elumalai, Nagarajan; Tavassoli, Ali; Firestein, Ron; Phoenix, Timothy N; D'Alessandro, Angelo; Dasgupta, Biplab

A Phase 0/I Pharmacokinetic and Pharmacodynamics and Safety and Tolerability Study of Letrozole in Combination with Standard Therapy in Recurrent High-Grade Gliomas

一项评估来曲唑联合标准疗法治疗复发性高级别胶质瘤的0/I期药代动力学、药效学、安全性和耐受性的研究

Desai, Pankaj B; Karve, Aniruddha S; Zawit, Misam; Arora, Priyanka; Dave, Nimita; Awosika, Joy; Li, Ningjing; Fuhrman, Bethany; Medvedovic, Mario; Sallans, Larry; Kendler, Ady; DasGupta, Biplab; Plas, David; Curry, Richard; Zuccarello, Mario; Chaudhary, Rekha; Sengupta, Soma; Wise-Draper, Trisha M

EXTH-99. SYSTEMIC AND BRAIN PHARMACOKINETICS OF A GABA(A) RECEPTOR AGONIST, AMLAL-101, AS AN INVESTIGATIONAL THERAPEUTIC FOR THE TREATMENT OF PRIMARY AND METASTATIC BRAIN CANCERS

EXTH-99. GABA(A)受体激动剂AMLAL-101作为治疗原发性和转移性脑癌的研究性疗法的全身和脑药代动力学

Hari, Riitta; Parkkonen, Lauri; Silva, David; Powell, Lyndsi; Kovacevich, Alexsandra; Pillai, Jagan A; Lynn, Audrey; Song, Sunah; Appleby, Brian S; Karve, Aniruddha; Ahmed, Taukir; Desai, Janki; Bhattacharya, Debanjan; Toukam, Donatien Kamdem; Gadgil, Sidharth; Pemberton, Merissa; Plas, David; Gudelsky, Gary; Sallans, Larry; Cook, James; Desai, Pankaj; Krummel, Daniel Pomeranz; Sengupta, Soma

Brain pharmacokinetics and metabolism of the AMP-activated protein kinase selective inhibitor SBI-0206965, an investigational agent for the treatment of glioblastoma

AMP 活化蛋白激酶选择性抑制剂 SBI-0206965(一种治疗胶质母细胞瘤的试验药物)的脑药代动力学和代谢

Janki M Desai, Aniruddha S Karve, Gary A Gudelsky, Mruniya V Gawali, William Seibel, Larry Sallans, Biplab DasGupta, Pankaj B Desai

Mechanisms of stearoyl CoA desaturase inhibitor sensitivity and acquired resistance in cancer

硬脂酰辅酶 A 去饱和酶抑制剂敏感性和癌症获得性耐药性的机制

Nicole Oatman, Nupur Dasgupta, Priyanka Arora, Kwangmin Choi, Mruniya V Gawali, Nishtha Gupta, Sreeja Parameswaran, Joseph Salomone, Julie A Reisz, Sean Lawler, Frank Furnari, Cameron Brennan, Jianqiang Wu, Larry Sallans, Gary Gudelsky, Pankaj Desai, Brian Gebelein, Matthew T Weirauch, Angelo D'Ales

Tocopherol controls D1 amino acid oxidation by oxygen radicals in Photosystem II

生育酚控制光系统II中氧自由基对D1氨基酸的氧化作用

Kumar, Aditya; Prasad, Ankush; Sedlářová, Michaela; Kale, Ravindra; Frankel, Laurie K; Sallans, Larry; Bricker, Terry M; Pospíšil, Pavel

Erratum for Mor et al., "Identification of a New Class of Antifungals Targeting the Synthesis of Fungal Sphingolipids"

Mor 等人的论文“鉴定一类靶向真菌鞘脂合成的新型抗真菌药物”的勘误

Mor, Visesato; Rella, Antonella; Farnoud, Amir M; Singh, Ashutosh; Munshi, Mansa; Bryan, Arielle; Naseem, Shamoon; Konopka, James B; Ojima, Iwao; Bullesbach, Erika; Ashbaugh, Alan; Linke, Michael J; Cushion, Melanie; Collins, Margaret; Ananthula, Hari Krishna; Sallans, Larry; Desai, Pankaj B; Wiederhold, Nathan P; Fothergill, Annette W; Kirkpatrick, William R; Patterson, Thomas; Wong, Lai Hong; Sinha, Sunita; Giaever, Guri; Nislow, Corey; Flaherty, Patrick; Pan, Xuewen; Cesar, Gabriele Vargas; de Melo Tavares, Patricia; Frases, Susana; Miranda, Kildare; Rodrigues, Marcio L; Luberto, Chiara; Nimrichter, Leonardo; Del Poeta, Maurizio

Preclinical pharmacokinetic evaluation to facilitate repurposing of tyrosine kinase inhibitors nilotinib and imatinib as antiviral agents

临床前药代动力学评估促进酪氨酸激酶抑制剂尼洛替尼和伊马替尼重新用作抗病毒药物

Hari Krishna Ananthula, Scott Parker, Erin Touchette, R Mark Buller, Gopi Patel, Daniel Kalman, Johanna S Salzer, Nadia Gallardo-Romero, Victoria Olson, Inger K Damon, Tessa Moir-Savitz, Larry Sallans, Milton H Werner, Catherine M Sherwin, Pankaj B Desai

Amino acid oxidation of the D1 and D2 proteins by oxygen radicals during photoinhibition of Photosystem II

光系统 II 的光抑制过程中氧自由基对 D1 和 D2 蛋白质进行氨基酸氧化

Ravindra Kale, Annette E Hebert, Laurie K Frankel, Larry Sallans, Terry M Bricker, Pavel Pospíšil

Use of protein cross-linking and radiolytic footprinting to elucidate PsbP and PsbQ interactions within higher plant Photosystem II

利用蛋白质交联和放射性足迹法阐明高等植物光系统II中PsbP和PsbQ的相互作用

Mummadisetti, Manjula P; Frankel, Laurie K; Bellamy, Henry D; Sallans, Larry; Goettert, Jost S; Brylinski, Michal; Limbach, Patrick A; Bricker, Terry M