日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Quantifying VMAT2 target occupancy at effective valbenazine doses and comparing to a novel VMAT2 inhibitor: a translational PET study

量化有效剂量缬苯那嗪下VMAT2靶点占有率并与新型VMAT2抑制剂进行比较:一项转化性PET研究

Terry-Lorenzo, Ryan; Albrecht, Daniel; Crouch, Sabrinia; Wong, Richard; Loewen, Gordon; Giri, Nagdeep; Skor, Heather; Lin, Kelly; Sandiego, Christine M; Pajonas, Meghan; Rabiner, Eugenii A; Gunn, Roger N; Russell, David S; Haubenberger, Dietrich

Cryptic and abundant marine viruses at the evolutionary origins of Earth's RNA virome

地球RNA病毒组进化起源中的隐秘而丰富的海洋病毒

Zayed, Ahmed A; Wainaina, James M; Dominguez-Huerta, Guillermo; Pelletier, Eric; Guo, Jiarong; Mohssen, Mohamed; Tian, Funing; Pratama, Akbar Adjie; Bolduc, Benjamin; Zablocki, Olivier; Cronin, Dylan; Solden, Lindsey; Delage, Erwan; Alberti, Adriana; Aury, Jean-Marc; Carradec, Quentin; da Silva, Corinne; Labadie, Karine; Poulain, Julie; Ruscheweyh, Hans-Joachim; Salazar, Guillem; Shatoff, Elan; Bundschuh, Ralf; Fredrick, Kurt; Kubatko, Laura S; Chaffron, Samuel; Culley, Alexander I; Sunagawa, Shinichi; Kuhn, Jens H; Wincker, Patrick; Sullivan, Matthew B; Acinas, Silvia G; Babin, Marcel; Bork, Peer; Boss, Emmanuel; Bowler, Chris; Cochrane, Guy; de Vargas, Colomban; Gorsky, Gabriel; Guidi, Lionel; Grimsley, Nigel; Hingamp, Pascal; Iudicone, Daniele; Jaillon, Olivier; Kandels, Stefanie; Karp-Boss, Lee; Karsenti, Eric; Not, Fabrice; Ogata, Hiroyuki; Poulton, Nicole; Pesant, Stéphane; Sardet, Christian; Speich, Sabrinia; Stemmann, Lars; Sullivan, Matthew B; Sungawa, Shinichi; Wincker, Patrick

Identification of GSK3186899/DDD853651 as a Preclinical Development Candidate for the Treatment of Visceral Leishmaniasis

确定 GSK3186899/DDD853651 为治疗内脏利什曼病的临床前开发候选药物

Thomas, Michael G; De Rycker, Manu; Ajakane, Myriam; Albrecht, Sébastian; Álvarez-Pedraglio, Ana Isabel; Boesche, Markus; Brand, Stephen; Campbell, Lorna; Cantizani-Perez, Juan; Cleghorn, Laura A T; Copley, Royston C B; Crouch, Sabrinia D; Daugan, Alain; Drewes, Gerard; Ferrer, Santiago; Ghidelli-Disse, Sonja; Gonzalez, Silvia; Gresham, Stephanie L; Hill, Alan P; Hindley, Sean J; Lowe, Rhiannon M; MacKenzie, Claire J; MacLean, Lorna; Manthri, Sujatha; Martin, Franck; Miguel-Siles, Juan; Nguyen, Van Loc; Norval, Suzanne; Osuna-Cabello, Maria; Woodland, Andrew; Patterson, Stephen; Pena, Imanol; Quesada-Campos, Maria Teresa; Reid, Iain H; Revill, Charlotte; Riley, Jennifer; Ruiz-Gomez, Jose Ramon; Shishikura, Yoko; Simeons, Frederick R C; Smith, Alasdair; Smith, Victoria C; Spinks, Daniel; Stojanovski, Laste; Thomas, John; Thompson, Stephen; Underwood, Tim; Gray, David W; Fiandor, Jose M; Gilbert, Ian H; Wyatt, Paul G; Read, Kevin D; Miles, Timothy J

Cyclin-dependent kinase 12 is a drug target for visceral leishmaniasis

细胞周期蛋白依赖性激酶12是内脏利什曼病的一种药物靶点。

Wyllie, Susan; Thomas, Michael; Patterson, Stephen; Crouch, Sabrinia; De Rycker, Manu; Lowe, Rhiannon; Gresham, Stephanie; Urbaniak, Michael D; Otto, Thomas D; Stojanovski, Laste; Simeons, Frederick R C; Manthri, Sujatha; MacLean, Lorna M; Zuccotto, Fabio; Homeyer, Nadine; Pflaumer, Hannah; Boesche, Markus; Sastry, Lalitha; Connolly, Paul; Albrecht, Sebastian; Berriman, Matt; Drewes, Gerard; Gray, David W; Ghidelli-Disse, Sonja; Dixon, Susan; Fiandor, Jose M; Wyatt, Paul G; Ferguson, Michael A J; Fairlamb, Alan H; Miles, Timothy J; Read, Kevin D; Gilbert, Ian H

Discovery and Optimization of 5-Amino-1,2,3-triazole-4-carboxamide Series against Trypanosoma cruzi

发现和优化 5-氨基-1,2,3-三唑-4-甲酰胺系列化合物对抗克氏锥虫

Brand, Stephen; Ko, Eun Jung; Viayna, Elisabet; Thompson, Stephen; Spinks, Daniel; Thomas, Michael; Sandberg, Lars; Francisco, Amanda F; Jayawardhana, Shiromani; Smith, Victoria C; Jansen, Chimed; De Rycker, Manu; Thomas, John; MacLean, Lorna; Osuna-Cabello, Maria; Riley, Jennifer; Scullion, Paul; Stojanovski, Laste; Simeons, Frederick R C; Epemolu, Ola; Shishikura, Yoko; Crouch, Sabrinia D; Bakshi, Tania S; Nixon, Christopher J; Reid, Iain H; Hill, Alan P; Underwood, Tim Z; Hindley, Sean J; Robinson, Sharon A; Kelly, John M; Fiandor, Jose M; Wyatt, Paul G; Marco, Maria; Miles, Timothy J; Read, Kevin D; Gilbert, Ian H

Identification and characterization of hundreds of potent and selective inhibitors of Trypanosoma brucei growth from a kinase-targeted library screening campaign

通过激酶靶向库筛选活动鉴定和表征数百种布氏锥虫生长的强效和选择性抑制剂

Rosario Diaz, Sandra A Luengo-Arratta, João D Seixas, Emanuele Amata, William Devine, Carlos Cordon-Obras, Domingo I Rojas-Barros, Elena Jimenez, Fatima Ortega, Sabrinia Crouch, Gonzalo Colmenarejo, Jose Maria Fiandor, Jose Julio Martin, Manuela Berlanga, Silvia Gonzalez, Pilar Manzano, Miguel Navar