日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Investigation of Potent Anti-Mycobacterium tuberculosis Agents Derived from Pyridine Derivatives Targeting the Enoyl Acyl Carrier Protein Reductase (InhA): Design, Synthesis, and Computational Analysis

靶向烯酰基载体蛋白还原酶(InhA)的吡啶衍生物高效抗结核分枝杆菌药物的研究:设计、合成和计算分析

Sabt, Ahmed; Korycka-Machala, Małgorzata; Kassem, Asmaa F; The Son, Ninh; Ha, Nguyen Xuan; Brzostek, Anna; Thabit, Mohamed G; Kawka, Malwina; Dziadek, Bożena; Elshamy, Abdelsamed I; Atwa, Ahmed M; Dziadek, Jarosław

Exploring the impact of the innovative compound 3-(3-(4-hydroxy-2-oxo-2H-chromen-3-yl)-5-(pyridin-3-yl)-1H-pyrazol-1-yl) indolin-2-one on accelerating wound recovery

探索创新化合物3-(3-(4-羟基-2-氧代-2H-色烯-3-基)-5-(吡啶-3-基)-1H-吡唑-1-基)吲哚啉-2-酮对加速伤口愈合的影响

Sabt, Ahmed; Abdelmegeed, Heba; Abdel-Razik, Abdel-Razik H; Thabit, Mohamed G; Balaha, Marwa; Shaldam, Moataz A; Reda, Ahmed M; Soliman, Ahmed A F; Abdelraof, Mohamed; Abdel Latif, Nehad A; Elghonemy, Mai M; Ahmed, Eman Y; Abdelrahman, Mohamed A; Batran, Rasha Z

STYK1 expression in breast cancer and its association with vascular invasion and clinicopathological features

STYK1在乳腺癌中的表达及其与血管侵犯和临床病理特征的关系

Mohammed, Rabab; Ismaeel, Amina; Alshaikh, Safa; Mubarak, Aalaa; Sabt, Sajedah; Selvam, Samvel

Design, synthesis, and molecular modeling of novel thiazolopyridine-based inhibitors of enoyl acyl carrier protein reductase (InhA) as anti-Mycobacterium tuberculosis agents

设计、合成和分子建模新型噻唑并吡啶类烯酰酰基载体蛋白还原酶(InhA)抑制剂作为抗结核分枝杆菌药物

Sabt, Ahmed; Korycka-Machała, Małgorzata; Kassem, Asmaa F; Saleh, Abdulrahman M; Farag, Hanaa; Shaldam, Moataz A; Thabit, Mohamed G; Brzostek, Anna; Kuzioła, Magdalena; Dziadek, Bożena; Ibrahim, Hoda Atef Abdelsattar; Lei, Xinsheng; Dziadek, Jarosław; Abdelrahman, Mohamed A

Vitreous hemorrhage in a patient on tirzepatide: Coincidence or drug induced?

服用替拉帕肽的患者出现玻璃体出血:是巧合还是药物诱发?

Azeem, Sitara; Bulushi, Lujain Al; Sabt, Buthaina Isa

Discovery of N'-(1-(coumarin-3-yl)ethylidene)benzenesulfonohydrazide as a novel wound healing enhancer: synthesis, biological assessment, and molecular modeling

发现 N'-(1-(香豆素-3-基)亚乙基)苯磺酰肼作为一种新型伤口愈合促进剂:合成、生物学评价和分子建模

Khaleel, Eman F; Abdelmegeed, Heba; Abdel-Razik, Abdel-Razik H; Ebaid, Manal S; Son, Ninh The; Ha, Nguyen Xuan; Atef Abdelsattar Ibrahim, Hoda; Abdelrahman, Mohamed A; Elshamy, Abdelsamed I; Dziadek, Jarosław; Sabt, Ahmed; Eldehna, Wagdy M

Design, synthesis, and biological assessment of a novel series of coumarin-tethered thiazole derivatives as potential antibacterial agents

设计、合成并生物学评价一系列新型香豆素连接的噻唑衍生物作为潜在抗菌剂

Ebaid, Manal S; Farag, Hanaa; Abdelraof, Mohamed; Saleh, Abdulrahman M; Thabit, Mohamed G; Dziadek, Jarosław; Youssef, Ahmed A; Sabt, Ahmed

Recent studies on protein kinase signaling inhibitors based on thiazoles: review to date

基于噻唑类化合物的蛋白激酶信号通路抑制剂的最新研究进展:综述

Ebaid, Manal S; Abdelsattar Ibrahim, Hoda Atef; Kassem, Asmaa F; Sabt, Ahmed

Benzenesulfonohydrazide-tethered non-fused and fused heterocycles as potential anti-mycobacterial agents targeting enoyl acyl carrier protein reductase (InhA) with antibiofilm activity

苯磺酰肼连接的非稠合和稠合杂环化合物作为潜在的抗分枝杆菌药物,靶向烯酰酰基载体蛋白还原酶(InhA),具有抗生物膜活性。

Al-Warhi, Tarfah; Sabt, Ahmed; Korycka-Machala, Małgorzata; Kassem, Asmaa F; Shaldam, Moataz A; Ibrahim, Hoda Atef Abdelsattar; Kawka, Malwina; Dziadek, Bożena; Kuzioła, Magdalena; Eldehna, Wagdy M; Dziadek, Jarosław

New pyrazolylindolin-2-one based coumarin derivatives as anti-melanoma agents: design, synthesis, dual BRAFV600E/VEGFR-2 inhibition, and computational studies

新型吡唑啉-2-酮类香豆素衍生物作为抗黑色素瘤药物:设计、合成、双重 BRAFV600E/VEGFR-2 抑制和计算研究

Ahmed Sabt, Mohammed A Khedr, Wagdy M Eldehna, Abdelsamed I Elshamy, Mohamed F Abdelhameed, Rasha M Allam, Rasha Z Batran