日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

New Insights into Bitopic Orthosteric/Allosteric Ligands of Cannabinoid Receptor Type 2

对 2 型大麻素受体双位正构/变构配体的新见解

Rebecca Ferrisi, Beatrice Polini, Caterina Ricardi, Francesca Gado, Kawthar A Mohamed, Giovanna Baron, Salvatore Faiella, Giulio Poli, Simona Rapposelli, Giuseppe Saccomanni, Giancarlo Aldini, Grazia Chiellini, Robert B Laprairie, Clementina Manera, Gabriella Ortore

Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: from Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands

新型 CB2 受体配体的设计、合成和生物活性:从正构和变构调节剂到双立体/双位配体

Francesca Gado, Rebecca Ferrisi, Beatrice Polini, Kawthar A Mohamed, Caterina Ricardi, Elena Lucarini, Sara Carpi, Federica Domenichini, Lesley A Stevenson, Simona Rapposelli, Giuseppe Saccomanni, Paola Nieri, Gabriella Ortore, Roger G Pertwee, Carla Ghelardini, Lorenzo Di Cesare Mannelli, Grazia Ch

Synthesis and In Vitro Characterization of Selective Cannabinoid CB2 Receptor Agonists: Biological Evaluation against Neuroblastoma Cancer Cells

选择性大麻素 CB2 受体激动剂的合成及体外表征:针对神经母细胞瘤癌细胞的生物学评价

Francesca Gado, Rebecca Ferrisi, Sarah Di Somma, Fabiana Napolitano, Kawthar A Mohamed, Lesley A Stevenson, Simona Rapposelli, Giuseppe Saccomanni, Giuseppe Portella, Roger G Pertwee, Robert B Laprairie, Anna Maria Malfitano, Clementina Manera

Design, synthesis and biological evaluation of novel orthosteric-allosteric ligands of the cannabinoid receptor type 2 (CB2R)

大麻素受体 2 型(CB2R)新型正构-变构配体的设计、合成及生物学评价

Rebecca Ferrisi, Francesca Gado, Beatrice Polini, Caterina Ricardi, Kawthar A Mohamed, Lesley A Stevenson, Gabriella Ortore, Simona Rapposelli, Giuseppe Saccomanni, Roger G Pertwee, Robert B Laprairie, Clementina Manera, Grazia Chiellini

Design, Synthesis, and In Vitro Evaluation of Novel 8-Amino-Quinoline Combined with Natural Antioxidant Acids

新型 8-氨基喹啉与天然抗氧化酸结合的设计、合成及体外评价

Andrea Bacci, Francesca Corsi, Massimiliano Runfola, Simona Sestito, Ilaria Piano, Clementina Manera, Giuseppe Saccomanni, Claudia Gargini, Simona Rapposelli

CB2-selective cannabinoid receptor ligands: synthesis, pharmacological evaluation, and molecular modeling investigation of 1,8-Naphthyridin-2(1H)-one-3-carboxamides

CB2 选择性大麻素受体配体:1,8-萘啶-2(1H)-酮-3-甲酰胺的合成、药理评价及分子建模研究

Valentina Lucchesi, Dow P Hurst, Derek M Shore, Simone Bertini, Brandie M Ehrmann, Marco Allarà, Lyle Lawrence, Alessia Ligresti, Filippo Minutolo, Giuseppe Saccomanni, Haleli Sharir, Marco Macchia, Vincenzo Di Marzo, Mary E Abood, Patricia H Reggio, Clementina Manera

Effects on immune cells of a new 1,8-naphthyridin-2-one derivative and its analogues as selective CB2 agonists: implications in multiple sclerosis

一种新型1,8-萘啶-2-酮衍生物及其类似物作为选择性CB2激动剂对免疫细胞的影响:在多发性硬化症中的意义

Malfitano, Anna Maria; Laezza, Chiara; D'Alessandro, Alba; Procaccini, Claudio; Saccomanni, Giuseppe; Tuccinardi, Tiziano; Manera, Clementina; Macchia, Marco; Matarese, Giuseppe; Gazzerro, Patrizia; Bifulco, Maurizio

Early outcome of arthroscopic Bankart's repair for recurrent traumatic anterior shoulder instability

关节镜下Bankart修复术治疗复发性创伤性前肩关节不稳的早期疗效

Saccomanni, Bernardino

A new test for acromio-clavicolar pathology

肩锁关节病理学的新检测方法

Saccomanni, Bernardino

Erratum to: Osteoid osteoma and osteoblastoma of the spine: a review of the literature

勘误:脊柱骨样骨瘤和成骨细胞瘤:文献综述

Saccomanni, Bernardino