日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Orthosteric STING inhibition elucidates molecular correction of SAVI STING.

正构 STING 抑制阐明了 SAVI STING 的分子矫正

Xie Tao, Ruzanov Max, Critton David, Merselis Leidy, Naglich Joseph, Sack John S, Zhang Ping, Xie Chunshan, Tredup Jeffrey, Stine Laurel B, Messier Cameron, Hope David L, Caceres-Cortes Janet, Mueller Luciano, Dyckman Alaric J, Newitt John A, Choudhury Asmita, Wilson Stephen C

X-ray structure of a human cardiac muscle troponin C/troponin I chimera in two crystal forms

人类心肌肌钙蛋白C/肌钙蛋白I嵌合体的两种晶体形式的X射线结构

Yan, Chunhong; Sack, John S

Azatricyclic Inverse Agonists of RORγt That Demonstrate Efficacy in Models of Rheumatoid Arthritis and Psoriasis

在类风湿性关节炎和银屑病模型中显示出疗效的RORγt氮杂三环反向激动剂

Liu, Qingjie; Xiao, Hai-Yun; Batt, Douglas G; Xiao, Zili; Zhu, Yeheng; Yang, Michael G; Li, Ning; Yip, Shiuhang; Li, Peng; Sun, Dawn; Wu, Dauh-Rurng; Ruzanov, Max; Sack, John S; Weigelt, Carolyn A; Wang, Jinhong; Li, Sha; Shuster, David J; Xie, Jenny H; Song, Yunling; Sherry, Tara; Obermeier, Mary T; Fura, Aberra; Stefanski, Kevin; Cornelius, Georgia; Chacko, Silvi; Khandelwal, Purnima; Dudhgaonkar, Shailesh; Rudra, Anjuman; Nagar, Jignesh; Murali, Venkata; Govindarajan, Arun; Denton, Rex; Zhao, Qihong; Meanwell, Nicholas A; Borzilleri, Robert; Dhar, T G Murali

Crystal structure of microtubule affinity-regulating kinase 4 catalytic domain in complex with a pyrazolopyrimidine inhibitor

微管亲和力调节激酶4催化结构域与吡唑并嘧啶抑制剂复合物的晶体结构

Sack, John S; Gao, Mian; Kiefer, Susan E; Myers, Joseph E Jr; Newitt, John A; Wu, Sophie; Yan, Chunhong

Discovery of a Highly Selective JAK2 Inhibitor, BMS-911543, for the Treatment of Myeloproliferative Neoplasms

发现一种高选择性JAK2抑制剂BMS-911543,用于治疗骨髓增生性肿瘤

Wan, Honghe; Schroeder, Gretchen M; Hart, Amy C; Inghrim, Jennifer; Grebinski, James; Tokarski, John S; Lorenzi, Matthew V; You, Dan; Mcdevitt, Theresa; Penhallow, Becky; Vuppugalla, Ragini; Zhang, Yueping; Gu, Xiaomei; Iyer, Ramaswamy; Lombardo, Louis J; Trainor, George L; Ruepp, Stefan; Lippy, Jonathan; Blat, Yuval; Sack, John S; Khan, Javed A; Stefanski, Kevin; Sleczka, Bogdan; Mathur, Arvind; Sun, Jung-Hui; Wong, Michael K; Wu, Dauh-Rurng; Li, Peng; Gupta, Anuradha; Arunachalam, P N; Pragalathan, Bala; Narayanan, Sankara; K C, Nanjundaswamy; Kuppusamy, Prakasam; Purandare, Ashok V