日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Kv2/Kv6.4 heteromeric potassium channels are expressed in spinal motor neurons and localized at C-bouton synapses

Kv2/Kv6.4异源钾通道在脊髓运动神经元中表达,并定位于C端突触。

Lacey, Taylor A; Murray, Karl D; Trimmer, James S; Sack, Jon T; Ferns, Michael J

A Kv2 inhibitor combination reveals native neuronal conductances consistent with Kv2/KvS heteromers

Kv2抑制剂组合揭示了与Kv2/KvS异聚体一致的天然神经元电导

Stewart, Robert G; Marquis, Matthew J; Jo, Sooyeon; Harris, Brandon; Aberra, Aman; Cook, Verity; Whiddon, Zachary; Yarov-Yarovoy, Vladimir; Ferns, Michael; Sack, Jon T

Structural modeling of hERG channel-drug interactions using Rosetta

利用 Rosetta 对 hERG 通道-药物相互作用进行结构建模

Emigh Cortez, Aiyana M; DeMarco, Kevin R; Furutani, Kazuharu; Bekker, Slava; Sack, Jon T; Wulff, Heike; Clancy, Colleen E; Vorobyov, Igor; Yarov-Yarovoy, Vladimir

K(+) takes the crown: Selective activation of non-selective crown ether channels

K(+) 占据主导地位:非选择性冠醚通道的选择性激活

Sack, Jon T

Pore opening, not voltage sensor movement, underpins the voltage-dependence of facilitation by a hERG blocker

hERG阻滞剂促进作用的电压依赖性是由孔隙开放而非电压传感器移动所致。

Furutani, Kazuharu; Kawano, Ryotaro; Ichiwara, Minami; Adachi, Ryo; Clancy, Colleen E; Sack, Jon T; Kita, Satomi

Molecular determinants of pro-arrhythmia proclivity of d- and l-sotalol via a multi-scale modeling pipeline

通过多尺度建模流程研究d-和l-索他洛尔致心律失常倾向的分子决定因素

DeMarco, Kevin R; Yang, Pei-Chi; Singh, Vikrant; Furutani, Kazuharu; Dawson, John R D; Jeng, Mao-Tsuen; Fettinger, James C; Bekker, Slava; Ngo, Van A; Noskov, Sergei Y; Yarov-Yarovoy, Vladimir; Sack, Jon T; Wulff, Heike; Clancy, Colleen E; Vorobyov, Igor

The tarantula toxin GxTx detains K(+) channel gating charges in their resting conformation

狼蛛毒素GxTx能使K(+)通道的门控电荷保持在静息构象。

Tilley, Drew C; Angueyra, Juan M; Eum, Kenneth S; Kim, Heesoo; Chao, Luke H; Peng, Anthony W; Sack, Jon T

Azide-Alkyne Click Conjugation on Quantum Dots by Selective Copper Coordination

通过选择性铜配位在量子点上实现叠氮-炔点击共轭

Mann, Victor R; Powers, Alexander S; Tilley, Drew C; Sack, Jon T; Cohen, Bruce E

Remodeling neuronal ER-PM junctions is a conserved nonconducting function of Kv2 plasma membrane ion channels.

重塑神经元内质网-质膜连接是 Kv2 质膜离子通道的保守非传导功能

Kirmiz Michael, Palacio Stephanie, Thapa Parashar, King Anna N, Sack Jon T, Trimmer James S

Tarantula toxins use common surfaces for interacting with Kv and ASIC ion channels

狼蛛毒素利用共同的表面与Kv和ASIC离子通道相互作用。

Gupta, Kanchan; Zamanian, Maryam; Bae, Chanhyung; Milescu, Mirela; Krepkiy, Dmitriy; Tilley, Drew C; Sack, Jon T; Yarov-Yarovoy, Vladimir; Kim, Jae Il; Swartz, Kenton J