Selective inhibition of the K(ir)2 family of inward rectifier potassium channels by a small molecule probe: the discovery, SAR, and pharmacological characterization of ML133
小分子探针对内向整流钾通道 K(ir)2 家族的选择性抑制:ML133 的发现、SAR 和药理学表征
期刊:ACS Chemical Biology
影响因子:3.5
doi:10.1021/cb200146a
Hao-Ran Wang, Meng Wu, Haibo Yu, Shunyou Long, Amy Stevens, Darren W Engers, Henry Sackin, J Scott Daniels, Eric S Dawson, Corey R Hopkins, Craig W Lindsley, Min Li, Owen B McManus