日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, synthesis, and anticancer activity of novel isocryptolepine 'aza' type acyl thiourea derivatives via combined experimental and computational approach

通过实验和计算相结合的方法设计、合成新型异隐花碱“氮杂”型酰基硫脲衍生物及其抗癌活性

Fayyaz, Ammara; Ejaz, Syeda Abida; Ahmed, Atteeque; Channar, Pervaiz Ali; Afzal, Saira; Ujan, Rabail; Saeed, Aamer; Bibi, Rifhat; Alsfouk, Bshra A; Abbas, Qamar; Sahito, Reshma; Bolte, Michael; Hökelek, Tuncer

Synthesis, characterization, in vitro and in silico studies of novel lophine clubbed acylthioureas

新型洛芬簇状酰基硫脲的合成、表征、体外和计算机模拟研究

Ullah, Sayyed Aqib; Jabeen, Hafsa; Javed, Areeba; Manan, Abdul; Irshad, Nadeem; Khan, Kashif Maqbool; Khushal, Aneela; Khan, Sara; Farooq, Umar; Bashir, Kashif; Saeed, Aamer

Deciphering the Anti-LUAD Mechanism of 4′-Demethyl-epipodophyllotoxin (4′-DMEP) via Machine Learning-Driven Target Identification and In Vitro Validation

利用机器学习驱动的靶点识别和体外验证,揭示4′-去甲基表鬼臼毒素(4′-DMEP)的抗肺腺癌机制

Lu, Jingwei; Aggarwal, Reeva; Pompili, Vincent J; Das, Hiranmoy; Chang, Wei; Yu, Jingjing; Di Palma, Roberto; Falco, Luigi; Coccia, Armando; Amitrano, Federica; D'Addio, Giovanni; La Rovere, Maria Teresa; Zhang, Yifang; Bao, Cuiping; Liu, Lingling; Liu, Renjiao; Wang, Xincheng; Guo, Xiaoxuan; Li, Chunjun; Wan, Qiliang; Ding, Yi; Liu, Wenduo; Yang, Kun; Zhang, Yue; Bu, Yifan; Song, Mingrong; Hao, Zhihua; Chen, Jing; Ouro, Alberto; Ben-Dor, Gabriel A; Debasa-Mouce, Manuel; Gulkarov, Shelly; De Leon, Joshua; Castro-Mosquera, Mónica; Sobrino, Tomás; Bougea, Anastasia; Reiss, Allison B; Szőke, Henrik; Vagedes, Jan; Balogh, Anikó; Li, Shengnian; Yin, Yikun; Guan, Jingjun; Yu, Liang; Jin, Shihao; Hu, Haotian; Wang, Xue; Wei, Xuan; Wang, Changjie; Ding, Peisen; Fan, Pengfei; Gao, Sinan; Dou, Xiaojing; Wang, Bing; Ma, Haoran; Yan, Mengwen; Liu, Jun; Zhu, Chen; Soria-Fregozo, Cesar; Ramos de Robles, Silvia Lizette; Flores-Soto, Mario Eduardo; Rosas-Sánchez, Gilberto Uriel; Zhao, Yannan; Deng, Bei; Li, Xiang; Zhang, Sheng; Chen, Yuhang; Peng, Dezhong; Sun, Ning; He, Yi; Liu, Yi-Wei; Chen, Gang-Lin; Chen, Lei; Yang, Hui-Lin; Lu, Jing-Kang; Xiong, Jing; Xiong, Xiao-Yi; He, Cheng-Qi; Barnett, Carlton C; Oliver, Gavin R; Schoenberg, Michael Rutenberg; Smith, Hans P; Smythe, W Roy; Zhang, Lei; Lu, Hao; Zhou, Hao; Bigjahan, Bavrina; Cavallari, Michele; Barisano, Giuseppe; Lange, Martin; Martinasek, Mary; Heckert, Nadine; Duan, Tingting; Zou, Changwei; Yang, Ming; Xu, Jiangxingzi; Wu, Zhaoping; Ullah, Sayyed Aqib; Jabeen, Hafsa; Javed, Areeba; Manan, Abdul; Irshad, Nadeem; Khan, Kashif Maqbool; Khushal, Aneela; Khan, Sara; Farooq, Umar; Bashir, Kashif; Saeed, Aamer; Cole, Paige L; Stead, Connor A; Burniston, Jatin G; Owens, Daniel J; Karnati, Bharath V; Kumar Behera, Pradip; Tripathy, Krishna P; Karanam, Rama Sowmya; Priyadarshini, Aparajita; Das, Swati; Mishra, Subhashree; Treiber, Kyle; Svensson, Robert; Cui, Zhong-lei; Zhang, Wen-hao; Wang, Wei; Han, Shan-shan; Zhu, Sai; Xu, Chuan-yi; Huang, Hua-sheng; Luo, Rong-hai; Pinky, Humayra Afroz; Nishan, MD Nahid Hassan; Alam, Gazi Md Ehsanul; Pathak, Ranjana; Goel, Anjana; Mukherjee, Archana; Patil, Deepali; Zope, Mukesh Kumar; Raj, Rishi; Devi, Seema; Bufacchi, Antonella; Pasciuti, Katia; Tesfaye, Melaku; Baheretibeb, Yonas; Dinku, Tsimona; Mihretu, Awoke; Li, Jie; Wang, Qiao-Yan; Xu, Xin; Cui, Lili; Zhang, Yong; Gu, Jingkai; Behboodi, Hamid-Reza; Asghari-Moghadam, Morteza; Mehri, Mehran; Hamza Ilyas, Muhammad; Daher, Mohammad; Deshpande, Viraj; Lindsay, Adam; Abboud, Joseph A; Kassam, Hafiz F; Yang, Runyu; Feng, Hui; Zhang, Mengyao; Liu, Yi; Luo, Minna; Liu, Ruimin; Wang, Kaiyao; Li, Qijing; Wang, Wenjuan; Chen, Jing; Du, Yue; Xiao, Jiayi; Yang, Bingyu; Niu, Fan; He, Pengcheng; Takahashi, Momo; Tamura, Yuma; Tamiya, Hajime; Terashima, Masato; Takahashi, Harunori; Banba, Nobuyuki; Nakatani, Yuki; Otani, Naoyuki; Ueno, Asuka; Yasu, Takanori; Maejima, Yasuhiro; Liu, Xin; Woo, Sukyung; Elemosho, Abdulaziz; Malekzadeh, Hamid; Kluemper, Jude C; Janis, Jeffrey E; Li, Yanxian; Sang, Jun; Li, Xuemei; Ding, Wenjing; Yang, Chunyan; Yang, Zheng; Zhao, Shiping; Liu, Yanfang; Cardoso, Barbara R; Steele, Euridice Martinez; Brayner, Barbara; Yuan, Xinyi; Bransby, Lisa; Cummins, Hannah; Lim, Yen Ying; Machado, Priscila; Liu, Qiang; Liu, Cui; Qin, Xin; Baba, Ainain; Baba, Obair Yousuf; Ahmad, Abid; Shahid, Misbah; Cho, Hyo-Moon; Le, Minh-Thi-Tuyet; Shin, Ji-Hye; Mai, Van-Hieu; Choi, Seri; An, Jin-Pyo; Lee, Yun-Sil; Oh, Won-Keun; Feng, Fang; Choi, Jihye; Ahn, Dohyun; Truong, Thi My Tien; Yim, Kyung June; Kim, Hyun-Jin; Jung, Man-Young; Lee, Hae-Won; Kim, Dong-Shin; Kang, Inhae; Zhao, Yi; Ai, Wei; Zhao, Jieyu; Yang, Xi; Liu, Wencheng; Ma, Yaru; Mou, Jianrui; Hai, Ao; Ji, Ran; Gan, Yu; Miao, Zhuang; Hu, Shilong; Huang, Zhenbo; Liu, Jin; Liu, Xianggen; Yang, Jun; Ke, Bowen; Khatib, Hasan; Ellsworth, Elijah; Badhwar, Norisha; Zuñiga-Eulogio, Miriam; Quinteros, Michael; Hernández-Moreno, Alberto; Hernández-Moreno, Tadeo; Sharma, Tapan; Olea-Flores, Monserrat; Ordóñez, Mario; Coste-Sanchez, Carla; Padilla-Benavides, Teresita; Navarro-Tito, Napoleón; Lohawittayanan, Duangporn; Khulmanee, Tachin; Thima, Kanthinich; Chabang, Napason; Yenjai, Wanchalerm; Kanjanasirirat, Phongthon; Schlaeppi, Patrick; Tantivess, Varisa; Phumisithikul, Tanadej; Ratcha-in, Detchart; Chotsriluecha, Sanisorn; Chuchaisuwannasri, Dhanita; Phanchana, Matthew; Pinthong, Nattapon; Patrapuvich, Rapatbhorn; Charoensutthivarakul, Sitthivut; Haakonde, Richard; Zyambo, Golden; Changula, Katendi; Mwenechanya, Roy; Muzandu, Kaampwe Mayovu; Mondal, Kalyan; Mandal, Abhijit; Vijay, Anuj; Patel, Ganeshkumar; Gong, Shan; Liu, Yeqian; Chen, Chunming; Feng, Min; Yang, Meiqi; Ren, Weiqiong; Wang, Min; Zhao, Shaojie; Yuan, Hua; Zhao, Min; Hang, Chen; Yuan, Rong; Canal de Velasco, Luis M; González Flores, José Emiliano; Kraus Fischer, Gabriel; Morales Arteaga, Jose Luis; Olivares Casas, María J; Alvarez Nava, Kenia N; Morales Morales, Frida M; Zhao, Tian-Pei; Chen, Jing-Yu; Li, Yue-Hua; Zhang, Chen-Xia; Ma, Yu-Xiang; Qin, Zhao; Wang, Xue-De; Liu, Hua-Min; Cui, Rui-Fu; Wang, Lei; Xu, Yong-Jun; Shi, Hai-Ming; Iizuka, Yusuke; Kosaka, Takuya; Kishi, Takahiro; Mitsuoka, Hiroshi; Yamaguchi, Yuki; Hoshino, Akihiro; Masuda, Hidemichi; Zhou, Xuchang; Wang, Dongxue; Deng, Huili; Guo, Jianmin; Chen, Xier; Lin, Zhangyu; Liu, Baolong; Zhao, Ruobing; Gao, Lu; Yin, Xuan; Zhang, Yun; Chen, Yan; Yang, Yajing; Li, Qingxian; Shen, Qu; Ji, Jianguang; Ni, Guoxin; Abikar, Apoorva; Ranganathan, Prathibha; Mottin, Melina; Jurisch, Christopher D; Silva-Mendonça, Sabrina; Seanego, Donald; Ramos, Paulo R P da Silva; Freitas, Caroline S; Mattos, Mayara; Fintelman-Rodrigues, Natalia; Sacramento, Carolina Q; Guivel-Benhassine, Florence; Bruel, Timothée; Krugmann, Liezl; Puhl, Ana C; Urbina, Fabio; Lane, Thomas R; Merten, Eric M; Pearce, Kenneth H; Lepioshkin, Alexander; Poromov, Artem; Monakhova, Natalia; Schwartz, Olivier; Chibale, Kelly; Souza, Thiago M L; Ekins, Sean; Makarov, Vadim; Gessner, Richard K; Andrade, Carolina H; Liang, Hui; Huang, Qinhong; Xian, Mingming; Chen, Taoliang; Sun, Xinlin; Binorkar, Sandeep V; Sawant, Ranjeet; Ukey, Rashtrapal N; Bhat, Ravindra; Monteblanco, Carlo D; Sy Su, Karl Matthew C; Jose, Geraldine Raphaela B; Yao, Jinghui; Wang, Chenhao; Wang, Zhichao; Xiang, Shi; Sun, Wu; Chen, Hui; Yang, Chao

Correction: Novel pyrimidine linked acyl thiourea derivatives as potent α-amylase and proteinase K inhibitors: design, synthesis, molecular docking and ADME studies

更正:新型嘧啶连接的酰基硫脲衍生物作为强效α-淀粉酶和蛋白酶K抑制剂:设计、合成、分子对接和ADME研究

Zaman, Hina; Saeed, Aamer; Ismail, Hammad; Anwaar, Sadaf; Latif, Muhammad; Hashmi, Muhammad Zaffar; El-Seedi, Hesham R

Three decades of selective product formation via Griesbaum co-ozonolysis: insight and advances (1995-2025)

格里斯鲍姆共臭氧分解选择性产物形成三十年:见解与进展(1995-2025)

Zain-Ul-Abideen, Muhammad; Saeed, Aamer; Haider, Mian Bilal; Shabir, Ghulam; El-Seedi, Hesham R

Exploration of novel triazolo-thiadiazine hybrids of deferasirox as multi-target-directed anti-neuroinflammatory agents with structure-activity relationship (SAR): a new treatment opportunity for Alzheimer's disease.

探索新型三唑噻二嗪杂合物地拉罗司作为多靶点导向抗神经炎症药物的结构活性关系(SAR):阿尔茨海默病的新治疗机会

Shakir Syed Ahmed, Rashid Umer, Marryum, Fatima Nighat, Ejaz Syeda Abida, Fayyaz Ammara, Ullah Muhammad Zahid, Saeed Aamer, Khan Ajmal, Al Harrasi Ahmed, Mumtaz Amara

Synthesis and evaluation of thiazolyl coumarin drug conjugates as carbonic anhydrase isozyme inhibitors by using integrated invitro and insilico approaches

利用体外和计算机模拟相结合的方法合成和评价噻唑基香豆素药物偶联物作为碳酸酐酶同工酶抑制剂的活性

Ahmed, Atteeque; Kanwal, Romaisa; Channar, Pervaiz Ali; Alshahrani, Mohammad Y; Saeed, Aamer; Ejaz, Syeda Abida; Attaullah, Hafiz Muhammad; Bibi, Rifhat; Li, Chen

Discovery of isatin-thiazole conjugates as potent urease inhibitors; synthesis, biochemical screening and computational studies

发现靛红-噻唑缀合物作为强效脲酶抑制剂;合成、生化筛选和计算研究

Haider, Mian Bilal; Zaib, Sumera; Saeed, Aamer; Ahmed, Atteeque; Javed, Hira; Areeba; Shabir, Ghulam; Irfan, Madiha; Othman, Gehan Ahmed

Ectonucleotidase inhibitors: targeting signaling pathways for therapeutic advancement-an in-depth review

外核苷酸酶抑制剂:靶向信号通路以推进治疗进展——深度综述

Sharafat, R Huzaifa; Saeed, Aamer

Novel pyrazoline linked acyl thiourea pharmacophores as antimicrobial, urease, amylase and α-glucosidase inhibitors: design, synthesis, SAR and molecular docking studies

新型吡唑啉连接的酰基硫脲药效团作为抗菌、脲酶、淀粉酶和α-葡萄糖苷酶抑制剂:设计、合成、构效关系和分子对接研究

Saeed, Aamer; Ahmed, Atteeque; Haider, Main Bilal; Ismail, Hammad; Hayat, Khizar; Shabir, Ghulam; El-Seedi, Hesham R