日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design and Evaluation of Andrographolide Analogues as SARS-CoV-2 Main Protease Inhibitors: Molecular Modeling and in vitro Studies

穿心莲内酯类似物作为SARS-CoV-2主蛋白酶抑制剂的设计与评价:分子建模和体外研究

Suriya, Utid; Intamalee, Pansachon; Saeeng, Rungnapha; Wilasluck, Patcharin; Deetanya, Peerapon; Wangkanont, Kittikhun; Kanjanasirirat, Phongthon; Wongwitayasombat, Chanikarn; Nutho, Bodee

Design and Synthesis of Mycophenolic Acid Analogues for Osteosarcoma Cancer Treatment.

设计并合成霉酚酸类似物用于骨肉瘤治疗

Silalai Patamawadee, Teeyakasem Pimpisa, Pruksakorn Dumnoensun, Saeeng Rungnapha

Piperine Enhances Mitochondrial Biogenesis to Mitigate Stress in SH-SY5Y Neuroblastoma Cells.

胡椒碱增强线粒体生物合成以减轻 SH-SY5Y 神经母细胞瘤细胞的应激反应

Saikachain Nongluk, Charoensawat Pawitchaya, Tuntoolavest Oramon, Vejsureeyakul Napak, Kunpittaya Teeranart, Poolsri Wanangkan, Sungkaworn Titiwat, Saeeng Rungnapha, Muanprasat Chatchai, Asavapanumas Nithi

Discovery of C-12 dithiocarbamate andrographolide analogue as a novel antioxidant and α-glucosidase inhibitors: In vitro and in silico studies

发现C-12二硫代氨基甲酸酯穿心莲内酯类似物作为新型抗氧化剂和α-葡萄糖苷酶抑制剂:体外和计算机模拟研究

Suriya, Utid; Duangtha, Chanathip; Dontricharoen, Thanchanok; Yamanont, Paveena; Kuhaudomlarp, Sakonwan; Thitiyanuwat, Prawit; Nutho, Bodee; Arsakhant, Patcharee; Saeeng, Rungnapha; Morales, Noppawan Phumala; Mangmool, Supachoke; Likitnukul, Sutharinee

siRNA Targeting Mcl-1 Potentiates the Anticancer Activity of Andrographolide Nanosuspensions via Apoptosis in Breast Cancer Cells

针对 Mcl-1 的 siRNA 通过诱导乳腺癌细胞凋亡增强穿心莲内酯纳米混悬液的抗癌活性

Supusson Pengnam, Purin Charoensuksai, Boon-Ek Yingyongnarongkul, Rungnapha Saeeng, Hasan Uludağ, Prasopchai Patrojanasophon, Praneet Opanasopit, Samarwadee Plianwong

Discovery of C-12 dithiocarbamate andrographolide analogues as inhibitors of SARS-CoV-2 main protease: In vitro and in silico studies

发现C-12二硫代氨基甲酸酯穿心莲内酯类似物作为SARS-CoV-2主蛋白酶抑制剂:体外和计算机模拟研究

Nutho, Bodee; Wilasluck, Patcharin; Deetanya, Peerapon; Wangkanont, Kittikhun; Arsakhant, Patcharee; Saeeng, Rungnapha; Rungrotmongkol, Thanyada

Antitumor effect of acanthoic acid against primary effusion lymphoma via inhibition of c-FLIP

棘酸通过抑制 c-FLIP 对原发性渗出性淋巴瘤发挥抗肿瘤作用

Gunya Sittithumcharee, Ryusho Kariya, Teerapich Kasemsuk, Rungnapha Saeeng, Seiji Okada

The anti-cancer activity of an andrographolide analogue functions through a GSK-3β-independent Wnt/β-catenin signaling pathway in colorectal cancer cells

穿心莲内酯类似物的抗癌活性是通过不依赖于 GSK-3β 的 Wnt/β-catenin 信号通路在结直肠癌细胞中发挥作用的。

Reabroi, Somrudee; Saeeng, Rungnapha; Boonmuen, Nittaya; Kasemsuk, Teerapich; Saengsawang, Witchuda; Suksen, Kanoknetr; Zhu, Weiming; Piyachaturawat, Pawinee; Chairoungdua, Arthit

Inhibition of Topoisomerase IIα and Induction of Apoptosis in Gastric Cancer Cells by 19-Triisopropyl Andrographolide

19-三异丙基穿心莲内酯抑制拓扑异构酶IIα并诱导胃癌细胞凋亡

Monger, Adeep; Boonmuen, Nittaya; Suksen, Kanoknetr; Saeeng, Rungnapha; Kasemsuk, Teerapich; Piyachaturawat, Pawinee; Saengsawang, Witchuda; Chairoungdua, Arthit