日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fluorescent Isostere (Fluostere) of the Carboxylate: Design of hDHODH Fluorescent Inhibitors as Proof of Concept

羧酸盐的荧光等排体(Fluostere):hDHODH荧光抑制剂的设计及其概念验证

Sainas, Stefano; Martino, Elena; Garino, Claudio; Circosta, Paola; Luganini, Anna; Giorgis, Marta; Bavo, Francesco; Piccinini, Marco; Ramondetti, Cristina; Alberti, Marta; Miggiano, Riccardo; Gribaudo, Giorgio; Boschi, Donatella; Frølund, Bente; Lolli, Marco Lucio

Expanding the MR1 ligandome using chemical class-specific fragmentation and molecular networking

利用化学类别特异性片段化和分子网络扩展MR1配体组

Lecchi, Chiara; Vacchini, Alessandro; Sainas, Stefano; Lolli, Marco L; Luedtke, Matthew; Mori, Lucia; De Libero, Gennaro; Balbo, Silvia; Villalta, Peter W

Radiosynthesis of [18F]brequinar for in vivo PET imaging of hDHODH for potential studies of acute myeloid leukemia and cancers

放射合成 [18F] 布喹那,用于 hDHODH 的体内 PET 成像,可用于急性髓系白血病和癌症的潜在研究

Vinay Kumar Banka, Stefano Sainas, Elena Martino, Jiacheng Wang, Marco Lucio Lolli, Yu-Shin Ding

Dihydroorotate dehydrogenase inhibition reveals metabolic vulnerability in chronic myeloid leukemia

二氢乳清酸脱氢酶抑制揭示慢性粒细胞白血病的代谢脆弱性

Mohammad Houshmand, Nicoletta Vitale #, Francesca Orso #, Alessandro Cignetti, Ivan Molineris, Valentina Gaidano, Stefano Sainas, Marta Giorgis, Donatella Boschi, Carmen Fava, Alice Passoni, Marta Gai, Massimo Geuna, Federica Sora, Alessandra Iurlo, Elisabetta Abruzzese, Massimo Breccia, Olga Mulas,

Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5- a]pyridine Scaffold: SAR of the Aryloxyaryl Moiety

使用基于 2-羟基吡唑并 [1,5- a] 吡啶骨架的强效人类二氢乳清酸脱氢酶抑制剂靶向治疗急性髓性白血病:芳氧基芳基部分的 SAR

Stefano Sainas, Marta Giorgis, Paola Circosta, Giulio Poli, Marta Alberti, Alice Passoni, Valentina Gaidano, Agnese C Pippione, Nicoletta Vitale, Davide Bonanni, Barbara Rolando, Alessandro Cignetti, Cristina Ramondetti, Alessia Lanno, Davide M Ferraris, Barbara Canepa, Barbara Buccinnà, Marco Picci

The Novel h DHODH Inhibitor MEDS433 Prevents Influenza Virus Replication by Blocking Pyrimidine Biosynthesis

新型 h DHODH 抑制剂 MEDS433 通过阻断嘧啶生物合成来阻止流感病毒复制

Giulia Sibille, Anna Luganini, Stefano Sainas, Donatella Boschi, Marco Lucio Lolli, Giorgio Gribaudo

Association between High Normal TSH Levels and Obesity in Women with Anti-Thyroid Autoantibodies (ATAs)

甲状腺抗抗体(ATA)阳性女性中高正常TSH水平与肥胖之间的关联

Velluzzi, Fernanda; Pisanu, Silvia; Galletta, Maura; Fosci, Michele; Secci, Gianni; Deledda, Andrea; Boi, Francesco; Rodia, Rossella; Fanciulli, Giuseppe; Delitala, Alessandro Palmerio; Sainas, Gianmarco; Loviselli, Andrea

Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2-Hydroxypyrazolo[1,5- a]pyridine Scaffold: SAR of the Biphenyl Moiety

使用基于 2-羟基吡唑并 [1,5- a] 吡啶骨架的强效人类二氢乳清酸脱氢酶抑制剂靶向治疗急性髓性白血病:联苯部分的 SAR

Stefano Sainas, Marta Giorgis, Paola Circosta, Valentina Gaidano, Davide Bonanni, Agnese C Pippione, Renzo Bagnati, Alice Passoni, Yaqi Qiu, Carina Florina Cojocaru, Barbara Canepa, Alessandro Bona, Barbara Rolando, Mariia Mishina, Cristina Ramondetti, Barbara Buccinnà, Marco Piccinini, Mohammad Hou

The New Generation h DHODH Inhibitor MEDS433 Hinders the In Vitro Replication of SARS-CoV-2 and Other Human Coronaviruses

新一代 h DHODH 抑制剂 MEDS433 可抑制 SARS-CoV-2 和其他人类冠状病毒的体外复制

Arianna Calistri, Anna Luganini, Barbara Mognetti, Elizabeth Elder, Giulia Sibille, Valeria Conciatori, Claudia Del Vecchio, Stefano Sainas, Donatella Boschi, Nuria Montserrat, Ali Mirazimi, Marco Lucio Lolli, Giorgio Gribaudo, Cristina Parolin

Systolic and Diastolic Functions After a Brief Acute Bout of Mild Exercise in Normobaric Hypoxia

常压低氧条件下短暂轻度运动后的收缩和舒张功能

Magnani, Sara; Mulliri, Gabriele; Roberto, Silvana; Sechi, Fabio; Ghiani, Giovanna; Sainas, Gianmarco; Nughedu, Giorgio; Vargiu, Romina; Bassareo, Pier Paolo; Crisafulli, Antonio