日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-based design of an opioid receptor modulator for enhanced morphine analgesia

基于结构的阿片受体调节剂设计及其在增强吗啡镇痛中的应用

Wang, Yue; Luo, Ping; Xu, Haiyan; Zhan, Li; Sakamoto, Kensuke; Li, Mingyu; Wang, Jing; Huang, Xi-Ping; Zhou, Jianhui; Liu, Tao; Suo, Yanrui; Fan, Wenjia; He, Xinheng; Xu, Youwei; Cai, Yongjie; Wang, Chao; Zhao, Yuxi; Dai, Antao; Lai, Yali; Yuan, Qingning; Hu, Wen; Wu, Kai; Yang, Dehua; Cheng, Xi; Lu, Xiaojie; Krumm, Brian; Kenakin, Terry; Zhang, Jian; Roth, Bryan L; Gao, Zhaobing; Xu, H Eric; Zhuang, Youwen

Large Library Docking for Polypharmacology

用于多药理学的大型库对接

Wu, Yujin; Vigneron, Seth; Braz, Joao; Srinivasan, Karthik; Fink, Elissa A; Huang, Xi-Ping; Xu, Xinyu; Huebner, Harald; Kim, Joseph Y; Wang, Jing; Pfeiffer, Tara; Sakamoto, Kensuke; Radchenko, Dmytro S; Rodriguiz, Ramona M; Moroz, Yurii S; Irwin, John J; Gmeiner, Peter; Billesboelle, Christian; Roth, Bryan L; Basbaum, Allan I; Manglik, Aashish; Wetsel, William C; Shoichet, Brian K

Cryo-EM Structures of Brain-Derived G Protein-Coupled Receptors: The First Direct Visualization from Mammalian Brain Tissue

脑源性G蛋白偶联受体的冷冻电镜结构:首次从哺乳动物脑组织中直接观察

Wright, Nicholas J; Chiu, Yi-Ting; Sakamoto, Kensuke; Kocak, D Dewran; Fordyce, Blake A; Hua, Kunjie; Huang, Karen Lu; Scherrer, Grégory; Lyons, Scott P; Roth, Bryan L

The selectivity implications of docking libraries with greater and lesser similarities to bio-like molecules

对接库与生物分子相似度高低的影响

Hall, Brendan W; Sakamoto, Kensuke; Huang, Xi-Ping; Irwin, John J; Shoichet, Brian K; Roth, Bryan L

AlphaFold2 structures guide prospective ligand discovery

AlphaFold2结构指导潜在配体的发现

Lyu, Jiankun; Kapolka, Nicholas; Gumpper, Ryan; Alon, Assaf; Wang, Liang; Jain, Manish K; Barros-Álvarez, Ximena; Sakamoto, Kensuke; Kim, Yoojoong; DiBerto, Jeffrey; Kim, Kuglae; Glenn, Isabella S; Tummino, Tia A; Huang, Sijie; Irwin, John J; Tarkhanova, Olga O; Moroz, Yurii; Skiniotis, Georgios; Kruse, Andrew C; Shoichet, Brian K; Roth, Bryan L

Structure-guided design of a peripherally restricted chemogenetic system.

结构导向的外周限制性化学遗传系统设计

Kang Hye Jin, Krumm Brian E, Tassou Adrien, Geron Matan, DiBerto Jeffrey F, Kapolka Nicholas J, Gumpper Ryan H, Sakamoto Kensuke, Dewran Kocak D, Olsen Reid H J, Huang Xi-Ping, Zhang Shicheng, Huang Karen L, Zaidi Saheem A, Nguyen MyV T, Jo Min Jeong, Katritch Vsevolod, Fay Jonathan F, Scherrer Grégory, Roth Bryan L

A comprehensive review of the genetic and biological evidence supports a role for MicroRNA-137 in the etiology of schizophrenia

对遗传学和生物学证据的全面回顾支持MicroRNA-137在精神分裂症病因学中的作用。

Sakamoto, Kensuke; Crowley, James J

miRNA-132: a dynamic regulator of cognitive capacity

miRNA-132:认知能力的动态调节因子

Hansen, Katelin F; Karelina, Kate; Sakamoto, Kensuke; Wayman, Gary A; Impey, Soren; Obrietan, Karl

MicroRNAs: a potential interface between the circadian clock and human health

微小RNA:生物钟与人类健康之间潜在的桥梁

Hansen, Katelin F; Sakamoto, Kensuke; Obrietan, Karl

Transcriptional regulation of ferritin and antioxidant genes by HIPK2 under genotoxic stress

基因毒性应激下HIPK2对铁蛋白和抗氧化基因的转录调控

Hailemariam, Kiros; Iwasaki, Kenta; Huang, Bo-Wen; Sakamoto, Kensuke; Tsuji, Yoshiaki