日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fexinidazole and Corallopyronin A target Wolbachia-infected sheath cells present in filarial nematodes

非西尼达唑和珊瑚吡喃酮A靶向丝状线虫中存在的沃尔巴克氏体感染的鞘细胞

Chappell, Laura; Peguero, Ricardo; Conner, William R; Fowler, Sommer; Cooper, Brandon S; Pfarr, Kenneth; Hoerauf, Achim; Lustigman, Sara; Sakanari, Judy; Sullivan, William

Fexinidazole and Corallopyronin A target Wolbachia-infected sheath cells present in filarial nematodes.

菲西尼达唑和珊瑚吡喃酮 A 靶向丝状线虫中存在的沃尔巴克氏体感染的鞘细胞

Chappell Laura, Peguero Ricardo, Conner William R, Fowler Sommer, Cooper Brandon, Pfarr Kenneth, Hoerauf Achim, Lustigman Sara, Sakanari Judy, Sullivan William

Repurposed Drugs That Activate Autophagy in Filarial Worms Act as Effective Macrofilaricides

激活丝虫自噬的再利用药物可作为有效的大丝虫杀虫剂

Denis Voronin, Nancy Tricoche, Ricardo Peguero, Anna Maria Kaminska, Elodie Ghedin, Judy A Sakanari, Sara Lustigman

Combinations of the azaquinazoline anti-Wolbachia agent, AWZ1066S, with benzimidazole anthelmintics synergise to mediate sub-seven-day sterilising and curative efficacies in experimental models of filariasis

抗沃尔巴克氏体药物AWZ1066S(一种氮杂喹唑啉类药物)与苯并咪唑类驱虫药联合使用,可产生协同作用,在丝虫病实验模型中于7天内达到灭菌和治愈效果。

Hegde, Shrilakshmi; Marriott, Amy E; Pionnier, Nicolas; Steven, Andrew; Bulman, Christina; Gunderson, Emma; Vogel, Ian; Koschel, Marianne; Ehrens, Alexandra; Lustigman, Sara; Voronin, Denis; Tricoche, Nancy; Hoerauf, Achim; Hübner, Marc P; Sakanari, Judy; Aljayyoussi, Ghaith; Gusovsky, Fabian; Dagley, Jessica; Hong, David W; O'Neill, Paul; Ward, Steven A; Taylor, Mark J; Turner, Joseph D

Antifungal and Antiparasitic Activities of Metallocene-Containing Fluconazole Derivatives

含茂金属的氟康唑衍生物的抗真菌和抗寄生虫活性

Lin, Yan; Scalese, Gonzalo; Bulman, Christina A; Vinck, Robin; Blacque, Olivier; Paulino, Margot; Ballesteros-Casallas, Andres; Pérez Díaz, Leticia; Salinas, Gustavo; Mitreva, Makedonka; Weil, Tobias; Cariou, Kevin; Sakanari, Judy A; Gambino, Dinorah; Gasser, Gilles

Uncovering the essential roles of glutamate carboxypeptidase 2 orthologs in Caenorhabditis elegans

揭示谷氨酸羧肽酶 2 直系同源物在秀丽隐杆线虫中的重要作用

Lucie Panska #, Stepanka Nedvedova #, Vojtech Vacek, Daniela Krivska, Lukas Konecny, Filip Knop, Zsofia Kutil, Lubica Skultetyova, Adrian Leontovyc, Lenka Ulrychova, Judy Sakanari, Masako Asahina, Cyril Barinka, Marie Macurkova, Jan Dvorak

Discovery of New Broad-Spectrum Anti-Infectives for Eukaryotic Pathogens Using Bioorganometallic Chemistry

利用生物有机金属化学发现针对真核病原体的新型广谱抗感染药物

Lin, Yan; Jung, Hyeim; Bulman, Christina A; Ng, James; Vinck, Robin; O'Beirne, Cillian; Zhong, Shuai; Moser, Matthew S; Tricoche, Nancy; Peguero, Ricardo; Li, Robert W; Urban, Joseph F Jr; Le Pape, Patrice; Pagniez, Fabrice; Moretto, Marco; Weil, Tobias; Lustigman, Sara; Cariou, Kevin; Mitreva, Makedonka; Sakanari, Judy A; Gasser, Gilles

Development and validation of small animal models for onchocerciasis and loiasis microfilaricide discovery

用于发现盘尾丝虫病和罗阿丝虫病微丝虫杀灭剂的小动物模型的开发和验证

Rene Bilingwe Ayiseh, Glory Enjong Mbah, Elvis Monya, Emmanuel Menang Ndi, Judy Sakanari, Sara Lustigman, Fidelis Cho-Ngwa

Biochemical and structural characterizations of thioredoxin reductase selenoproteins of the parasitic filarial nematodes Brugia malayi and Onchocerca volvulus

寄生丝虫马来丝虫和盘尾丝虫的硫氧还蛋白还原酶硒蛋白的生化和结构特征

Francesca Fata, Radosveta Gencheva, Qing Cheng, Rachel Lullo, Matteo Ardini, Ilaria Silvestri, Federica Gabriele, Rodolfo Ippoliti, Christina A Bulman, Judy A Sakanari, David L Williams, Elias S J Arnér, Francesco Angelucci

Aspartyl Protease Inhibitors as Anti-Filarial Drugs

天冬氨酰蛋白酶抑制剂作为抗丝虫病药物

Liana Beld, Hyeim Jung, Christina A Bulman, Bruce A Rosa, Peter U Fischer, James W Janetka, Sara Lustigman, Judy A Sakanari, Makedonka Mitreva