日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Multi-layered molecular profiling informs the diagnosis and targeted therapy of desmoplastic small round cell tumor

多层分子谱分析为促纤维增生性小圆细胞肿瘤的诊断和靶向治疗提供信息

Renner, Marcus; Oleś, Małgorzata; Paramasivam, Nagarajan; Heilig, Christoph E; Schneider, Annika; Modugno, Caroline; Herremans, Catherine; Hüllein, Jennifer; Hutter, Barbara; Erkut, Cihan; Mock, Andreas; Krieghoff-Henning, Eva; Jensen, Cecilia B; Sakhteman, Amirhossein; The, Matthew; Prinz, Tony; Lajer, Panna; Baude-Müller, Annika; Beck, Katja; Beuthien-Baumann, Bettina; Apostolidis, Leonidas; Bauer, Sebastian; Boerries, Melanie; Brandts, Christian H; Rieke, Damian T; Kindler, Thomas; Klauschen, Frederick; Schulze-Osthoff, Klaus; Schlenk, Richard F; Berchem, Guy; Allgäuer, Michael; Mechtersheimer, Gunhild; Stenzinger, Albrecht; Lipka, Daniel B; Schlesner, Matthias; Kuster, Bernhard; Jahn, Arne; Schröck, Evelin; Heining, Christoph; Teleanu, Maria-Veronica; Horak, Peter; Kreutzfeldt, Simon; Hübschmann, Daniel; Hartmann, Wolfgang; Glimm, Hanno; Fröhling, Stefan

Mapping drug mechanisms with ProteomicsDB: unified omics and cell sensitivity data at scale

利用 ProteomicsDB 绘制药物机制图谱:大规模统一的组学和细胞敏感性数据

Picciani, Mario; Soleymaniniya, Armin; Müller, Julian; Sakhteman, Amirhossein; Tzanakis, Konstantinos; Bernett, Judith; Kahl, Elias; Hamood, Firas; Kersting, Johannes; Pourjam, Mohsen; Nagai, Luis Augusto Eijy; List, Markus; Kuster, Bernhard; The, Matthew; Wilhelm, Mathias

Decrypting the molecular basis of cellular drug phenotypes by dose-resolved expression proteomics

利用剂量分辨表达蛋白质组学揭示细胞药物表型的分子基础

Eckert, Stephan; Berner, Nicola; Kramer, Karl; Schneider, Annika; Müller, Julian; Lechner, Severin; Brajkovic, Sarah; Sakhteman, Amirhossein; Graetz, Christian; Fackler, Jonas; Dudek, Michael; Pfaffl, Michael W; Knolle, Percy; Wilhelm, Stephanie; Kuster, Bernhard

Gemcitabine and ATR inhibitors synergize to kill PDAC cells by blocking DNA damage response

吉西他滨和 ATR 抑制剂协同作用,通过阻断 DNA 损伤反应杀死 PDAC 细胞

Stefanie Höfer, Larissa Frasch, Sarah Brajkovic, Kerstin Putzker, Joe Lewis, Hendrik Schürmann, Valentina Leone, Amirhossein Sakhteman, Matthew The, Florian P Bayer, Julian Müller, Firas Hamood, Jens T Siveke, Maximilian Reichert, Bernhard Kuster

Serendipitous and Systematic Chemoproteomic Discovery of MBLAC2, HINT1, and NME1-4 Inhibitors from Histone Deacetylase-Targeting Pharmacophores

从组蛋白去乙酰化酶靶向药效团中偶然发现和系统性化学蛋白质组学方法鉴定 MBLAC2、HINT1 和 NME1-4 抑制剂

Lechner, Severin; Sha, Shuyao; Sethiya, Jigar Paras; Szczupak, Patrycja; Dolot, Rafal; Lomada, Santosh; Sakhteman, Amirhossein; Tushaus, Johanna; Prokofeva, Polina; Krauss, Michael; Breu, Ferdinand; Vögerl, Katharina; Morgenstern, Martin; Hrabě de Angelis, Martin; Haucke, Volker; Wieland, Thomas; Wagner, Carston; Médard, Guillaume; Bracher, Franz; Kuster, Bernhard

Illuminating phenotypic drug responses of sarcoma cells to kinase inhibitors by phosphoproteomics.

利用磷酸化蛋白质组学揭示肉瘤细胞对激酶抑制剂的表型药物反应

Lee Chien-Yun, The Matthew, Meng Chen, Bayer Florian P, Putzker Kerstin, Müller Julian, Streubel Johanna, Woortman Julia, Sakhteman Amirhossein, Resch Moritz, Schneider Annika, Wilhelm Stephanie, Kuster Bernhard

Decrypting lysine deacetylase inhibitor action and protein modifications by dose-resolved proteomics

通过剂量分辨蛋白质组学解密赖氨酸脱乙酰酶抑制剂作用和蛋白质修饰

Yun-Chien Chang, Christian Gnann, Raphael R Steimbach, Florian P Bayer, Severin Lechner, Amirhossein Sakhteman, Miriam Abele, Jana Zecha, Jakob Trendel, Matthew The, Emma Lundberg, Aubry K Miller, Bernhard Kuster

A combination of virtual screening, molecular dynamics simulation, MM/PBSA, ADMET, and DFT calculations to identify a potential DPP4 inhibitor

结合虚拟筛选、分子动力学模拟、MM/PBSA、ADMET 和 DFT 计算,以鉴定潜在的 DPP4 抑制剂

Zare, Fateme; Ataollahi, Elaheh; Mardaneh, Pegah; Sakhteman, Amirhossein; Keshavarz, Valiollah; Solhjoo, Aida; Emami, Leila

Correlation of Myeloid-Derived Suppressor Cell Expansion with Upregulated Transposable Elements in Severe COVID-19 Unveiled in Single-Cell RNA Sequencing Reanalysis

单细胞RNA测序再分析揭示重症COVID-19中髓系来源抑制细胞扩增与转座元件上调的相关性

Farahmandnejad, Mitra; Mosaddeghi, Pouria; Dorvash, Mohammadreza; Sakhteman, Amirhossein; Negahdaripour, Manica; Faridi, Pouya

A region-resolved proteomic map of the human brain enabled by high-throughput proteomics

利用高通量蛋白质组学技术构建人脑区域分辨蛋白质组图谱

Tüshaus, Johanna; Sakhteman, Amirhossein; Lechner, Severin; The, Matthew; Mucha, Eike; Krisp, Christoph; Schlegel, Jürgen; Delbridge, Claire; Kuster, Bernhard