日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An electrophilic fragment screening for the development of small molecules targeting caspase-2

亲电片段筛选用于开发针对 caspase-2 的小分子

Matthew E Cuellar, Mu Yang, Surendra Karavadhi, Ya-Qin Zhang, Hu Zhu, Hongmao Sun, Min Shen, Matthew D Hall, Samarjit Patnaik, Karen H Ashe, Michael A Walters, Steffen Pockes

Target Class Profiling of Small-Molecule Methyltransferases

小分子甲基转移酶的靶标类别分析

Quinlin M Hanson, Nate Hoxie, Min Shen, Hui Guo, Ig-Jun Cho, Ipsita Chakraborty, Brooklyn M Aragon, Ganesha Rai, Samarjit Patnaik, John S Janiszewski, Matthew D Hall

Ligand-Induced Activation of GPR110 (ADGRF1) to Improve Visual Function Impaired by Optic Nerve Injury

配体诱导激活 GPR110 (ADGRF1) 可改善视神经损伤导致的视觉功能障碍

Heung-Sun Kwon, Karl Kevala, Haohua Qian, Mones Abu-Asab, Samarjit Patnaik, Juan Marugan, Hee-Yong Kim

Upregulation of the ESCRT pathway and multivesicular bodies accelerates degradation of proteins associated with neurodegeneration

ESCRT 通路和多泡体的上调加速了与神经退行性疾病相关的蛋白质的降解

Ron Benyair, Sai Srinivas Panapakkam Giridharan, Pilar Rivero-Ríos, Junya Hasegawa, Emily Bristow, Eeva-Liisa Eskelinen, Merav D Shmueli, Vered Fishbain-Yoskovitz, Yifat Merbl, Lisa M Sharkey, Henry L Paulson, Phyllis I Hanson, Samarjit Patnaik, Ismael Al-Ramahi, Juan Botas, Juan Marugan, Lois S Wei

Discovery and Optimization of Pyrrolopyrimidine Derivatives as Selective Disruptors of the Perinucleolar Compartment, a Marker of Tumor Progression toward Metastasis

发现并优化吡咯并嘧啶衍生物作为核仁周围区室的选择性破坏剂(肿瘤向转移发展的标志)

Kevin J Frankowski, Samarjit Patnaik, Chen Wang, Noel Southall, Dipannita Dutta, Soumitta De, Dandan Li, Christopher Dextras, Yi-Han Lin, Marthe Bryant-Connah, Danielle Davis, Feijun Wang, Leah M Wachsmuth, Pranav Shah, Jordan Williams, Md Kabir, Edward Zhu, Bolormaa Baljinnyam, Amy Wang, Xin Xu, Jo

Discovery of Small-Molecule VapC1 Nuclease Inhibitors by Virtual Screening and Scaffold Hopping from an Atomic Structure Revealing Protein-Protein Interactions with a Native VapB1 Inhibitor

通过虚拟筛选和基于原子结构的骨架跃迁发现小分子VapC1核酸酶抑制剂,揭示其与天然VapB1抑制剂的蛋白质-蛋白质相互作用

Hongmao Sun,Nathan P Coussens,Carina Danchik,Leah M Wachsmuth,Mark J Henderson,Samarjit Patnaik,Matthew D Hall,Ashley L Molinaro,Dayle A Daines,Min Shen

Discovery of Novel Small-Molecule Scaffolds for the Inhibition and Activation of WIP1 Phosphatase from a RapidFire Mass Spectrometry High-Throughput Screen

通过 RapidFire 质谱高通量筛选发现用于抑制和激活 WIP1 磷酸酶的新型小分子支架

Victor Clausse, Yuhong Fang, Dingyin Tao, Harichandra D Tagad, Hongmao Sun, Yuhong Wang, Surendra Karavadhi, Kelly Lane, Zhen-Dan Shi, Olga Vasalatiy, Christopher A LeClair, Rebecca Eells, Min Shen, Samarjit Patnaik, Ettore Appella, Nathan P Coussens, Matthew D Hall, Daniel H Appella

Activation of mitochondrial TRAP1 stimulates mitochondria-lysosome crosstalk and correction of lysosomal dysfunction

线粒体 TRAP1 的激活可刺激线粒体-溶酶体串扰并纠正溶酶体功能障碍

Fannie W Chen, Joanna P Davies, Raul Calvo, Jagruti Chaudhari, Georgia Dolios, Mercedes K Taylor, Samarjit Patnaik, Jean Dehdashti, Rebecca Mull, Patricia Dranchack, Amy Wang, Xin Xu, Emma Hughes, Noel Southall, Marc Ferrer, Rong Wang, Juan J Marugan, Yiannis A Ioannou

The HIV protease inhibitor, ritonavir, corrects diverse brain phenotypes across development in mouse model of DYT-TOR1A dystonia

HIV 蛋白酶抑制剂利托那韦可纠正 DYT-TOR1A 肌张力障碍小鼠模型中发育过程中的各种大脑表型

Zachary F Caffall, Bradley J Wilkes, Ricardo Hernández-Martinez, Joseph E Rittiner, Jennifer T Fox, Kanny K Wan, Miranda K Shipman, Steven A Titus, Ya-Qin Zhang, Samarjit Patnaik, Matthew D Hall, Matthew B Boxer, Min Shen, Zhuyin Li, David E Vaillancourt, Nicole Calakos

Identification of Small Molecule Inhibitors of a Mir155 Transcriptional Reporter in Th17 Cells

Th17 细胞中 Mir155 转录报告基因的小分子抑制剂的鉴定

Anju Singh, Myagmarjav Dashynam, Bryan Chim, Thelma M Escobar, Xiuhuai Liu, Xin Hu, Samarjit Patnaik, Xin Xu, Noel Southall, Juan Marugan, Ajit Jadhav, Vanja Lazarevic, Stefan A Muljo, Marc Ferrer