MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants
MK-5172,一种选择性抑制丙型肝炎病毒NS3/4a蛋白酶的药物,对多种基因型和耐药变异株均具有广泛活性。
期刊:Antimicrobial Agents and Chemotherapy
影响因子:4.5
doi:10.1128/AAC.01066-13
Draper, Michael P; Weir, S; Macone, A; Donatelli, J; Trieber, C A; Tanaka, S K; Levy, Stuart B; P, Shahul Hameed; Solapure, Suresh; Mukherjee, Kakoli; Nandi, Vrinda; Waterson, David; Shandil, Radha; Balganesh, Meenakshi; Sambandamurthy, Vasan K; Raichurkar, Anand Kumar; Deshpande, Abhijeet; Ghosh, Anirban; Awasthy, Disha; Shanbhag, Gajanan; Sheikh, Gulebahar; McMiken, Helen; Puttur, Jayashree; Reddy, Jitendar; Werngren, Jim; Read, Jon; Kumar, Mahesh; R, Manjunatha; Chinnapattu, Murugan; Madhavapeddi, Prashanti; Manjrekar, Praveena; Basu, Reetobrata; Gaonkar, Sheshagiri; Sharma, Sreevalli; Hoffner, Sven; Humnabadkar, Vaishali; Subbulakshmi, Venkita; Panduga, Vijender; Summa, Vincenzo; Ludmerer, Steven W; McCauley, John A; Fandozzi, Christine; Burlein, Christine; Claudio, Giuliano; Coleman, Paul J; DiMuzio, Jillian M; Ferrara, Marco; Filippo, Marcello Di; Gates, Adam T; Graham, Donald J; Harper, Steven; Hazuda, Daria J; Huang, Qian; McHale, Carolyn; Monteagudo, Edith; Pucci, Vincenzo; Rowley, Michael; Rudd, Michael T; Soriano, Aileen; Stahlhut, Mark W; Vacca, Joseph P; Olsen, David B; Liverton, Nigel J; Carroll, Steven S