日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Menaquinone depletion resensitises bedaquiline-resistant tuberculosis

甲萘醌耗竭可使耐贝达喹啉结核病重新敏感

Wetzel, Jennefer; Dallow, John; Davis, Ellie; Pearson, William H; Daems, Stijn; Govaerts, Matthias; Hereijgers, Joyce; Sprangers, Joke; Truebody, Barry; Maes, Valerie; van Hasselt, Vera; Leemans, Annelies; Pujari, Venugopal; Vos, Ann; Viturro, Carlos M Martínez; Gómez, José Enrique; Peeters, Mirte; Gerber, Michelle; Chhabra, Nandini; Wouters, Annelies; Everaerts, Melissa; Painter, Hannah; Fathima, Raisha; Willcocks, Sam J; Davies, Cadi; Raeymaekers, Valerie; Clark, Taane G; Draghia-Akli, Ruxandra; Fletcher, Helen; Van Loock, Marnix; Hibberd, Martin L; Mostowy, Serge; Crick, Dean C; Pym, Alexander S; Samby, Kirandeep; Jackson, Paul; Trabanco, Andrés A; Larrouy-Maumus, Gerald; Steyn, Adrie J C; Stoops, Bart; Dhar, Neeraj; Aguilar-Pérez, Clara; Lamprecht, Dirk A; Wall, Richard J; Koul, Anil

Screening of Medicines for Malaria Venture Open Boxes Identifies Potent SARS-CoV‑2 Papain-like Protease (PL(pro)) Inhibitors

疟疾药物筛选项目“开放盒子”发现了强效的SARS-CoV-2木瓜蛋白酶样蛋白酶(PL(pro))抑制剂

Gawriljuk, Victor Oliveira; Noske, Gabriela Dias; Fernandes, Rafaela Sachetto; Nakamura, Aline Minalli; Freire, Marjorie C L C; Godoy, Mariana Ortiz; Bonatto, Vinicius; Chelucci, Rafael; Andricopulo, Adriano; Bakowski, Malina A; Wolff, Karen C; Riva, Laura; Burrows, Jeremy N; Wells, Timothy N C; Laleu, Benoît; Martins, Ronaldo; Souza, Juliano Paula; Arruda, Eurico; Samby, Kirandeep; Laskar, Sujay; Guido, Rafael Victorio Carvalho; Oliva, Glaucius; Godoy, Andre Schutzer

Global Health Priority Box─Proactive Pandemic Preparedness

全球卫生优先事项栏目——主动应对大流行病

Adam, Anna; Besson, Dominique; Bryant, Rob; Rees, Sarah; Willis, Paul A; Burrows, Jeremy N; Hooft van Huisjduijnen, Rob; Laleu, Benoît; Norton, Larry; Canan, Stacie; Hawryluk, Natalie; Robinson, Dale; Palmer, Mike; Samby, Kirandeep Kaur

Molnupiravir combined with different repurposed drugs further inhibits SARS-CoV-2 infection in human nasal epithelium in vitro

莫努匹拉韦与不同再利用药物联合使用可在体外进一步抑制人鼻腔上皮细胞中的 SARS-CoV-2 感染

Hulda R Jonsdottir, Denise Siegrist, Thomas Julien, Blandine Padey, Mendy Bouveret, Olivier Terrier, Andres Pizzorno, Song Huang, Kirandeep Samby, Timothy N C Wells, Bernadett Boda, Manuel Rosa-Calatrava, Olivier B Engler, Samuel Constant

Screening of the Pandemic Response Box Reveals an Association between Antifungal Effects of MMV1593537 and the Cell Wall of Cryptococcus neoformans, Cryptococcus deuterogattii, and Candida auris

对大流行病应对盒的筛选揭示了MMV1593537的抗真菌作用与新型隐球菌、德氏隐球菌和耳念珠菌细胞壁之间的关联

de Oliveira, Haroldo C; Castelli, Rafael F; Reis, Flavia C G; Samby, Kirandeep; Nosanchuk, Joshua D; Alves, Lysangela R; Rodrigues, Marcio L

The Antifungal Itraconazole Is a Potent Inhibitor of Chikungunya Virus Replication

抗真菌药物伊曲康唑是基孔肯雅病毒复制的强效抑制剂

Policastro, Lucca R; Dolci, Isabela; Godoy, Andre S; Silva Júnior, José V J; Ruiz, Uriel E A; Santos, Igor A; Jardim, Ana C G; Samby, Kirandeep; Burrows, Jeremy N; Wells, Timothy N C; Gil, Laura H V G; Oliva, Glaucius; Fernandes, Rafaela S

Screening the pandemic response box identified benzimidazole carbamates, Olorofim and ravuconazole as promising drug candidates for the treatment of eumycetoma

对疫情应对方案库的筛选发现,苯并咪唑氨基甲酸酯类化合物、奥洛芬和拉伏康唑是治疗真菌性足菌肿的潜在候选药物。

Lim, Wilson; Nyuykonge, Bertrand; Eadie, Kimberly; Konings, Mickey; Smeets, Juli; Fahal, Ahmed; Bonifaz, Alexandro; Todd, Matthew; Perry, Benjamin; Samby, Kirandeep; Burrows, Jeremy; Verbon, Annelies; van de Sande, Wendy

A High-Throughput Phenotypic Screen of the 'Pandemic Response Box' Identifies a Quinoline Derivative with Significant Anthelmintic Activity

“大流行反应盒”的高通量表型筛选鉴定出具有显著驱虫活性的喹啉衍生物

Harrison T Shanley, Aya C Taki, Joseph J Byrne, Abdul Jabbar, Tim N C Wells, Kirandeep Samby, Peter R Boag, Nghi Nguyen, Brad E Sleebs, Robin B Gasser

Barcoded Asaia bacteria enable mosquito in vivo screens and identify novel systemic insecticides and inhibitors of malaria transmission

条形码 Asaia 细菌可实现蚊子体内筛查,并识别新型系统性杀虫剂和疟疾传播抑制剂

Angelika Sturm, Martijn W Vos, Rob Henderson, Maarten Eldering, Karin M J Koolen, Avinash Sheshachalam, Guido Favia, Kirandeep Samby, Esperanza Herreros, Koen J Dechering

Drug repurposing screens reveal cell-type-specific entry pathways and FDA-approved drugs active against SARS-Cov-2

药物再利用筛选揭示细胞类型特异性进入途径和 FDA 批准的抗 SARS-Cov-2 药物

Mark Dittmar, Jae Seung Lee, Kanupriya Whig, Elisha Segrist, Minghua Li, Brinda Kamalia, Lauren Castellana, Kasirajan Ayyanathan, Fabian L Cardenas-Diaz, Edward E Morrisey, Rachel Truitt, Wenli Yang, Kellie Jurado, Kirandeep Samby, Holly Ramage, David C Schultz, Sara Cherry