日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Scalable Design for Proximity-Inducing Molecules

一种可扩展的邻近诱导分子设计

Karaj, Endri; Venkatarangan, Varsha; Sindi, Shaimaa H; Siriwongsup, Surached; Lee, Chaiheon; Pergu, Rajaiah; Sreekanth, Vedagopuram; Kailass, Karishma; Tran, Kien; Singh, Prashant; Singh, Sameek; Kawai, Junya; Fung, Jeffrey E; Tefera, Mahilet; Dhaliwal, Rohil; Chaudhary, Santosh K; Keyes, April; Sadagopan, Ananthan; Boatner, Lisa; Shah, Neel H; Fehl, Charlie; Backus, Keriann M; Choudhary, Amit

Phosphorylation-Inducing Molecules for Regulating Dynamic Cellular Processes

调控动态细胞过程的磷酸化诱导分子

Pergu, Rajaiah; Sreekanth, Vedagopuram; Kokkonda, Praveen; Lai, Sophia; Tiwari, Praveen K; Singh, Sameek; Kawai, Junya; Singha, Santanu; Tian, Wenzhi; Thimaradka, Vikram; Siriwongsup, Surached; Tran, Kien; Choudhary, Amit

Growth factor receptor plasticity drives therapeutic persistence of metastatic breast cancer

生长因子受体可塑性驱动转移性乳腺癌的治疗持久性

Ayers, Mitchell; Monteiro, Marvis; Kulkarni, Aneesha; Reeser, Julie W; Dykhuizen, Emily; Roychowdhury, Sameek; Wendt, Michael K

Prevalence and biological impact of clinically relevant gene fusions in head and neck cancers

头颈癌中具有临床意义的基因融合的患病率和生物学影响

Hoskins, Emily L; Vella, Raven; Reeser, Julie W; Wing, Michele R; Samorodnitsky, Eric; Turkoglu, Altan; Stein, Leah; Breuning, Elizabeth; Risch, Zachary A; Hernandez-Sanchez, Wilnelly M; Yu, Lianbo; Churchman, Michelle; Single, Nancy; Chahoud, Jad; Jimeno, Antonio; Cavnar, Michael J; Reilley, Matthew; Scaife, Courtney; Nepple, Kenneth G; Phan, Minh; Schneider, Bryan; Edge, Stephen; Salhia, Bodour; Leiser, Aliza; Wise-Draper, Trisha M; Wendt, Michael K; Roychowdhury, Sameek

Orthogonal resistance mechanisms of classical- and induced-proximity inhibitors.

经典邻近抑制剂和诱导邻近抑制剂的正交耐药机制

Merz Manuel L, Kailass Karishma, Pergu Rajaiah, Tran Kien, Gupta Kritika, Severance Zachary C, Singh Sameek, Vedagopuram Sreekanth, Law Benjamin K, Rosenblatt Gideon, Dhaliwal Rohil, Choudhary Amit

Phosphorylation-inducing chimera rewires oncogenic kinase to trigger apoptosis.

磷酸化诱导嵌合体重塑致癌激酶以触发细胞凋亡

Merz Manuel L, Shoba Veronika M, Pergu Rajaiah, Severance Zachary C, Munkanatta Godage Dhanushka N P, Deb Arghya, Kwok Hui Si, Singh Prashant, Singh Sameek, Allen Jonathan B, Tian Wenzhi, Gosavi Pallavi M, Chaudhary Santosh K, Anokhina Viktoriya, Weisberg Ellen L, Payne N Connor, He Yao, Osadchey Reilly, Shekhar Mrinal, Mazitschek Ralph, Rees Matthew G, Roth Jennifer A, Cui Qiang, Griffin James D, Liau Brian B, Choudhary Amit

FGFR2-fusions define a clinically actionable molecular subset of pancreatic cancer

FGFR2融合基因定义了胰腺癌中具有临床意义的分子亚型。

Stein, Leah; Murugesan, Karthikeyan; Reeser, Julie W; Risch, Zachary; Wing, Michele R; Paruchuri, Anoosha; Samorodnitsky, Eric; Hoskins, Emily L; Dao, Thuy; Smith, Amy; Le, Dat; Babcook, Melissa A; Chang, Yi Seok; Avenarius, Matthew R; Imam, Muhammad; Freud, Aharon G; Roychowdhury, Sameek

Myeloid neoplasm with histiocytosis and spleen tyrosine kinase fusion responds to fostamatinib

伴有组织细胞增生和脾酪氨酸激酶融合的髓系肿瘤对福斯他替尼有反应

Risch, Zachary; Kaffenberger, Benjamin H; Chung, Catherine G; Samorodnitsky, Eric; Hoskins, Emily L; Dao, Thuy; Smith, Amy; Wall, Sarah A; Brammer, Jonathan; Reeser, Julie W; Wing, Michele R; Hopkins, Julia F; Albacker, Lee A; Abruzzo, Lynne V; Eisele, Caprice D; Freud, Aharon G; Roychowdhury, Sameek; Walsh, Katherine E

Risk Factors Predicting Outcomes in Advanced Upper Gastrointestinal Cancers Treated With Immune Checkpoint Inhibitors

预测接受免疫检查点抑制剂治疗的晚期上消化道癌症患者预后的风险因素

Manne, Ashish; Tounkara, Fode; Min, Eric; Samuel, Paul; Benson, Katherine; Noonan, Anne M; Mittra, Arjun; Hays, John; Roychowdhury, Sameek; Malalur, Pannaga; Rahman, Shafia; Jin, Ning; Pitter, Kenneth; Miller, Eric; Diaz, Alexandra; He, Kai

Mature MUC5AC Expression in Resected Pancreatic Ductal Adenocarcinoma Predicts Treatment Response and Outcomes

切除的胰腺导管腺癌中成熟的 MUC5AC 表达可预测治疗反应和结果

Ashish Manne, Ashwini Esnakula, Ankur Sheel, Amir Sara, Upender Manne, Ravi Kumar Paluri, Kai He, Wancai Yang, Davendra Sohal, Anup Kasi, Anne M Noonan, Arjun Mittra, John Hays, Sameek Roychowdhury, Pannaga Malalur, Shafia Rahman, Ning Jin, Jordan M Cloyd, Susan Tsai, Aslam Ejaz, Kenneth Pitter, Eri