日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Oxa-noribogaine reduces alcohol drinking through aversion learning and by altering glutamatergic activity in the mPFC

奥沙-诺瑞博格碱通过厌恶学习和改变内侧前额叶皮层谷氨酸能活性来减少酒精摄入。

Meinhardt, Marcus; Skorodumov, Ivan; Walter, Florian; Akan, Merve; Buchborn, Tobias; Prieult, Yéléna LE; Urban, Marvin; Spanagel, Rainer; von Ammon, Livia; Hopf, Carsten; Kalinichenko, Liubov; Mueller, Christian; Winter, Christine; Hadar, Ravit; Gül, Asude Zülal; Massuda, Ben; Hildebrandt, Maj; Domi, Esi; Keshishian, Adana; Ciccocioppo, Roberto; Sames, Dalibor; Havel, Vaclav; Woods, Leah; Beeson, Angela

Seeing the Spikes: The Future of Targetable Synthetic Voltage Sensors

洞察尖峰:可靶向合成电压传感器的未来

Fiala, Tomas; Sulzer, David; Sames, Dalibor

Molecular Design of SERTlight: A Fluorescent Serotonin Probe for Neuronal Labeling in the Brain

SERTlight的分子设计:一种用于大脑神经元标记的荧光血清素探针

Lee, Wei-Li; Westergaard, Xavier; Hwu, Christopher; Hwu, Jennifer; Fiala, Tomas; Lacefield, Clay; Boltaev, Umed; Mendieta, Adriana M; Lin, Lisa; Sonders, Mark S; Brown, Keaon R; He, Keer; Asher, Wesley B; Javitch, Jonathan A; Sulzer, David; Sames, Dalibor

Pharmacological Mechanism of the Non-hallucinogenic 5-HT(2A) Agonist Ariadne and Analogs

非致幻性 5-HT(2A) 激动剂 Ariadne 及其类似物的药理机制

Cunningham, Michael J; Bock, Hailey A; Serrano, Inis C; Bechand, Benjamin; Vidyadhara, D J; Bonniwell, Emma M; Lankri, David; Duggan, Priscilla; Nazarova, Antonina L; Cao, Andrew B; Calkins, Maggie M; Khirsariya, Prashant; Hwu, Christopher; Katritch, Vsevolod; Chandra, Sreeganga S; McCorvy, John D; Sames, Dalibor

Site selective C-H functionalization of Mitragyna alkaloids reveals a molecular switch for tuning opioid receptor signaling efficacy

帽柱木碱的位点选择性CH官能化揭示了一种调节阿片受体信号传导效力的分子开关

Bhowmik, Srijita; Galeta, Juraj; Havel, Václav; Nelson, Melissa; Faouzi, Abdelfattah; Bechand, Benjamin; Ansonoff, Mike; Fiala, Tomas; Hunkele, Amanda; Kruegel, Andrew C; Pintar, John E; Majumdar, Susruta; Javitch, Jonathan A; Sames, Dalibor

Development of a Dual Fluorescent and Magnetic Resonance False Neurotransmitter That Reports Accumulation and Release from Dopaminergic Synaptic Vesicles

开发一种双重荧光和磁共振成像的假神经递质,用于报告多巴胺能突触囊泡的积累和释放

Post, Michael R; Lee, Wei-Li; Guo, Jia; Sames, Dalibor; Sulzer, David

Chemical Targeting of Voltage Sensitive Dyes to Specific Cells and Molecules in the Brain

利用化学方法将电压敏感染料靶向大脑中的特定细胞和分子

Fiala, Tomas; Wang, Jihang; Dunn, Matthew; Šebej, Peter; Choi, Se Joon; Nwadibia, Ekeoma C; Fialova, Eva; Martinez, Diana M; Cheetham, Claire E; Fogle, Keri J; Palladino, Michael J; Freyberg, Zachary; Sulzer, David; Sames, Dalibor

7-Hydroxymitragynine Is an Active Metabolite of Mitragynine and a Key Mediator of Its Analgesic Effects

7-羟基帽柱木碱是帽柱木碱的活性代谢产物,也是其镇痛作用的关键介质。

Kruegel, Andrew C; Uprety, Rajendra; Grinnell, Steven G; Langreck, Cory; Pekarskaya, Elizabeth A; Le Rouzic, Valerie; Ansonoff, Michael; Gassaway, Madalee M; Pintar, John E; Pasternak, Gavril W; Javitch, Jonathan A; Majumdar, Susruta; Sames, Dalibor

Toward Serotonin Fluorescent False Neurotransmitters: Development of Fluorescent Dual Serotonin and Vesicular Monoamine Transporter Substrates for Visualizing Serotonin Neurons

迈向血清素荧光假神经递质:开发用于可视化血清素神经元的荧光双重血清素和囊泡单胺转运体底物

Henke, Adam; Kovalyova, Yekaterina; Dunn, Matthew; Dreier, Dominik; Gubernator, Niko G; Dincheva, Iva; Hwu, Christopher; Šebej, Peter; Ansorge, Mark S; Sulzer, David; Sames, Dalibor

Identification of Fluorescent Small Molecule Compounds for Synaptic Labeling by Image-Based, High-Content Screening.

通过基于图像的高内涵筛选鉴定用于突触标记的荧光小分子化合物

Dunn Matthew, Boltaev Umed, Beskow Anne, Pampou Sergey, Realubit Ronald, Meira Torcato, Silva João Vaz, Reeb Rose, Karan Charles, Jockusch Steffen, Sulzer David, Chang Young Tae, Sames Dalibor, Waites Clarissa L