日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Bridging mechanism and design: modern medicinal chemistry approaches to thymidylate synthase inhibitors

桥接机制与设计:现代药物化学方法在胸苷酸合成酶抑制剂中的应用

Al-Karmalawy, Ahmed A; Eissa, Mohamed E; Yousef, Tarek A; Al Khatib, Arwa Omar; Hawas, Samia S

Targeting cell cycle and apoptotic pathways with newly synthesized diselenide-linked imidazolone analogues with strong CDK6-targeting potential

利用新合成的具有强 CDK6 靶向潜力的二硒化物连接的咪唑酮类似物靶向细胞周期和凋亡通路

Abdel-Motaal, Marwa; Shaaban, Saad; Hawas, Samia S; Elsharif, Asma M; Sharaky, Marwa; Alatawi, Fatema S; Eissa, Mohamed E; Al Khatib, Arwa Omar; Abd El-Lateef, Hany M; Asem, Medhat; Al-Karmalawy, Ahmed A

Hybrid benzylidene thiazolidine-2,4-diones as potent apoptosis-inducing anticancer agents: design-driven optimization, cytotoxic profiling, and mechanistic validation in prostate cancer

杂合亚苄基噻唑烷-2,4-二酮类化合物作为强效的凋亡诱导型抗癌药物:基于设计的优化、细胞毒性分析以及在前列腺癌中的机制验证

Shaaban, Saad; Hawas, Samia S; Sharaky, Marwa; Ba-Ghazal, Hussein; Elmaaty, Ayman Abo; Alomari, Khadra B; Alaasar, Mohamed; Elsharif, Asma M; Alatawi, Fatema S; Mohamed, Mohamed Alaa; Al Khatib, Arwa Omar; Al-Karmalawy, Ahmed A

Organoselenium-based Schiff bases and amidic acid derivatives as promising anticancer agents targeting breast cancer by downregulating BCL-2: design, synthesis, and biological evaluation

基于有机硒的席夫碱和酰胺酸衍生物作为靶向乳腺癌、通过下调BCL-2表达的潜在抗癌药物:设计、合成和生物学评价

Shaaban, Saad; Hawas, Samia S; Elsharif, Asma M; Sharaky, Marwa; Ba-Ghazal, Hussein; Alaasar, Mohamed; Alatawi, Fatema S; Alomari, Khadra B; Eissa, Mohamed E; Al Khatib, Arwa Omar; Alnajjar, Radwan; Al-Karmalawy, Ahmed A

Sequential biosorptive-degradative remediation of methylene blue from polluted soil and wastewater by a newly isolated Bacillus safensis SMAH biomass: optimization, kinetics, isotherms and thermodynamics assessments

利用新分离的枯草芽孢杆菌SMAH生物质对受污染土壤和废水中的亚甲基蓝进行顺序生物吸附-降解修复:优化、动力学、等温线和热力学评估

Mahmoud, Mohamed E; Moneer, Abeer A; Abouelkheir, Samia S; Abdelfattah, Mohamed T M; Abdel-Aal, Hany

In silico interaction analysis of selected natural compounds with bacteriophage-encoded hyaluronate lyase from Streptococcus pyogenes

利用计算机模拟分析选定的天然化合物与化脓性链球菌噬菌体编码的透明质酸裂解酶的相互作用

Alkhalil, Samia S

A Diagnostic Pitfall: Secondary Syphilis Mimicking Psoriasis in a Patient With Alcoholic Liver Disease

诊断陷阱:酒精性肝病患者二期梅毒酷似银屑病

Armstrong, Julia L; Rankin, Erica; Singh Shrestha, Prakriti; Siddiqui, Samia S; Turkistani, Arifa; Evora, Jorge E; Rodriguez Caballero, Inima; Ghandi-Patel, Arohi; Samaniego, Vanessa S; Rodriguez, Ivan D

Multi-Targeted Mechanisms of Phytochemicals in Mitigating Cadmium-Induced Breast Cancer

植物化学物质缓解镉诱导乳腺癌的多靶点机制

Fidudusola, Fidara F; Odewumi, Caroline O; Latinwo, Lekan M; Oguntunde, Oluwatobi A; Messeha, Samia S; Soliman, Karam F A

Nrf2 Activation as a Therapeutic Target for Flavonoids in Aging-Related Osteoporosis

Nrf2激活作为类黄酮治疗衰老相关骨质疏松症的靶点

Messeha, Samia S; Fidudusola, Fidara F; Gendy, Sherif; Latinwo, Lekan M; Odewumi, Caroline O; Soliman, Karam F A

Medicinal chemistry perspectives on anticancer drug design based on clinical applications (2015-2025)

基于临床应用的抗癌药物设计药物化学展望(2015-2025)

Al-Karmalawy, Ahmed A; Eissa, Mohamed E; Ashour, Nada A; Yousef, Tarek A; Al Khatib, Arwa Omar; Hawas, Samia S