日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of Novel JAK2 Inhibitors from Amino Derivatives of Epoxyalantolactone: In Silico and In Vitro Studies

从环氧阿兰内酯氨基衍生物中鉴定新型JAK2抑制剂:计算机模拟和体外研究

Todsaporn, Duangjai; Sanachai, Kamonpan; Aonbangkhen, Chanat; Poo-Arporn, Rungtiva P; Kartsev, Victor; Pukhov, Sergey; Afanasyeva, Svetlana; Geronikaki, Athina; Rungrotmongkol, Thanyada

Natural Product-Inspired Bis(trifluoromethyl) Phenyl Hydroxycinnamate Derivatives as Promising Nonsteroidal Inhibitors of Human Steroid 5α-Reductase Type-1: Synthesis, In Vitro, and In Silico Studies

天然产物启发的双(三氟甲基)苯基羟基肉桂酸酯衍生物作为有前景的人甾体5α-还原酶1型非甾体抑制剂:合成、体外和计算机模拟研究

Isswanich, Kulpornsorn; Poungcho, Pattara; Buaban, Koonchira; Chuntakaruk, Hathaichanok; Sanachai, Kamonpan; Chansriniyom, Chaisak; Rungrotmongkol, Thanyada; De-Eknamkul, Wanchai; Chamni, Supakarn

Exploring novel furochochicine derivatives as promising JAK2 inhibitors in HeLa cells: Integrating docking, QSAR-ML, MD simulations, and experiments.

探索新型呋喃妥因衍生物作为 HeLa 细胞中 JAK2 抑制剂的潜力:整合对接、QSAR-ML、MD 模拟和实验

Todsaporn Duangjai, Sanachai Kamonpan, Aonbangkhen Chanat, Geronikaki Athina, Kartsev Victor, Lichitsky Boris, Komogortsev Andrey, Maitarad Phornphimon, Rungrotmongkol Thanyada

Molecular and structural characterization of a novel β-hemoglobinopathy caused by in Cis β-globin mutations in a Thai individual

对一名泰国个体中由顺式β-珠蛋白突变引起的新型β-血红蛋白病进行分子和结构表征

Singha, Kritsada; Pansuwan, Anupong; Sanachai, Kamonpan; Nutho, Bodee; Fucharoen, Goonnapa; Fucharoen, Supan

Pharmacogenetics and Precision Medicine Approaches for the Improvement of COVID-19 Therapies

药物遗传学和精准医学方法在改善新冠肺炎治疗中的应用

Biswas, Mohitosh; Sawajan, Nares; Rungrotmongkol, Thanyada; Sanachai, Kamonpan; Ershadian, Maliheh; Sukasem, Chonlaphat

Two flavonoid-based compounds from Murraya paniculata as novel human carbonic anhydrase isozyme II inhibitors detected by a resazurin yeast-based assay

通过基于刃天青酵母的检测方法,从九里香中分离出两种黄酮类化合物,作为新型人碳酸酐酶同工酶II抑制剂。

Sangkaew, Anyaporn; Samritsakulchai, Nawara; Sanachai, Kamonpan; Rungrotmongkol, Thanyada; Chavasiri, Warinthorn; Yompakdee, Chulee