Optimal linker length for small molecule PROTACs that selectively target p38α and p38β for degradation
选择性靶向 p38α 和 p38β 进行降解的小分子 PROTAC 的最佳接头长度
期刊:European Journal of Medicinal Chemistry
影响因子:6
doi:10.1016/j.ejmech.2020.112451
Craig Donoghue, Monica Cubillos-Rojas, Nuria Gutierrez-Prat, Carolina Sanchez-Zarzalejo, Xavier Verdaguer, Antoni Riera, Angel R Nebreda