日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design of Bicyclic Peptide Tandems Mimicking the Homodimeric GDF15 Protein to Inhibit GDF15-GFRaL-RET Complex Cell Signaling

设计模拟同源二聚体GDF15蛋白的双环肽串联体以抑制GDF15-GFRaL-RET复合物细胞信号传导

Noisier, Anaïs F M; Sandmark, Jenny; Edfeldt, Fredrik; Backmark, Anna; Broddefalk, Johan; Wandzik, Joanna; Jurva, Ulrik; Ek, Margareta; Johansson, Carina A; Barlind, Louise; Gunnarsson, Jenny; Bigalke, Janna M; Xue, Yafeng; Frolov, Andrey I; Kankkonen, Cecilia; Roth, Robert G; Fritsch, Maria; Watcham, Sophie; van Rietschoten, Katerine; Mudd, Gemma E; Harrison, Helen; Chen, Liuhong; Skynner, Michael J; Craik, David J; Chankeshwara, Sunay V; Lemurell, Malin

Identification and analyses of inhibitors targeting apolipoprotein(a) kringle domains KIV-7, KIV-10, and KV provide insight into kringle domain function

鉴定和分析针对载脂蛋白 (a) 的 kringle 域 KIV-7、KIV-10 和 KV 的抑制剂,有助于深入了解 kringle 域的功能

Jenny Sandmark, Anna Tigerström, Tomas Akerud, Magnus Althage, Thomas Antonsson, Stefan Blaho, Cristian Bodin, Jonas Boström, Yantao Chen, Anders Dahlén, Per-Olof Eriksson, Emma Evertsson, Tomas Fex, Ola Fjellström, David Gustafsson, Margareta Herslöf, Ryan Hicks, Emelie Jarkvist, Carina Johansson, 

Cryo-EM structure of the activated RET signaling complex reveals the importance of its cysteine-rich domain

激活的 RET 信号复合物的低温电子显微镜结构揭示了其富含半胱氨酸的结构域的重要性

Janna M Bigalke, Shintaro Aibara, Robert Roth, Göran Dahl, Euan Gordon, Sarah Dorbéus, A Amunts, Jenny Sandmark

Structural analysis identifies an escape route from the adverse lipogenic effects of liver X receptor ligands

结构分析确定了避免肝脏 X 受体配体不利脂肪生成影响的途径

Anna Y Belorusova, Emma Evertsson, Daniel Hovdal, Jenny Sandmark, Emma Bratt, Ingela Maxvall, Ira G Schulman, Peter Åkerblad, Eva-Lotte Lindstedt

Design of Selective sPLA(2)-X Inhibitor (-)-2-{2-[Carbamoyl-6-(trifluoromethoxy)-1H-indol-1-yl]pyridine-2-yl}propanoic Acid

选择性 sPLA(2)-X 抑制剂 (-)-2-{2-[氨基甲酰基-6-(三氟甲氧基)-1H-吲哚-1-基]吡啶-2-基}丙酸的设计

Giordanetto, Fabrizio; Knerr, Laurent; Nordberg, Peter; Pettersen, Daniel; Selmi, Nidhal; Beisel, Hans-Georg; de la Motte, Hannah; Månsson, Åsa; Dahlström, Mikael; Broddefalk, Johan; Saarinen, Gabrielle; Klingegård, Fredrik; Hurt-Camejo, Eva; Rosengren, Birgitta; Wikström, Johannes; Wågberg, Maria; Brengdahl, Johan; Rohman, Mattias; Sandmark, Jenny; Åkerud, Tomas; Roth, Robert G; Jansen, Frank; Ahlqvist, Marie

Structure and biophysical characterization of the human full-length neurturin-GFRa2 complex: A role for heparan sulfate in signaling

人类全长神经营养因子-GFRa2复合物的结构和生物物理特性:硫酸肝素在信号传导中的作用

Jenny Sandmark, Göran Dahl, Linda Öster, Bingze Xu, Patrik Johansson, Tomas Akerud, Anna Aagaard, Pia Davidsson, Janna M Bigalke, Maria Sörhede Winzell, G Jonah Rainey, Robert G Roth

Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A(2) Type X (sPLA(2)-X) Inhibitors.

发现一系列吲哚-2 甲酰胺类化合物作为选择性分泌型磷脂酶 A(2) X 型 (sPLA(2)-X) 抑制剂

Knerr Laurent, Giordanetto Fabrizio, Nordberg Peter, Pettersen Daniel, Selmi Nidhal, Beisel Hans-Georg, de la Motte Hannah, Olsson Thomas, Perkins Tim D J, Herslöf Margareta, Månsson à sa, Dahlström Mikael, Starke Ingemar, Broddefalk Johan, Saarinen Gabrielle, Klingegård Fredrik, Hurt-Camejo Eva, Rosengren Birgitta, Brengdahl Johan, Jansen Frank, Rohman Mattias, Sandmark Jenny, Hallberg Kenth, à kerud Tomas, Roth Robert G, Ahlqvist Marie

Creating novel activated factor XI inhibitors through fragment based lead generation and structure aided drug design

通过基于片段的先导化合物生成和结构辅助药物设计创建新的活化因子 XI 抑制剂

Ola Fjellström, Sibel Akkaya, Hans-Georg Beisel, Per-Olof Eriksson, Karl Erixon, David Gustafsson, Ulrik Jurva, Daiwu Kang, David Karis, Wolfgang Knecht, Viveca Nerme, Ingemar Nilsson, Thomas Olsson, Alma Redzic, Robert Roth, Jenny Sandmark, Anna Tigerström, Linda Öster

Understanding long-term sick leave in female white-collar workers with burnout and stress-related diagnoses: a qualitative study

了解患有职业倦怠和压力相关疾病的女性白领员工的长期病假情况:一项定性研究

Sandmark, Hélène; Renstig, Monica

Osteoarthrosis of the knee in men and women in association with overweight, smoking, and hormone therapy

男性和女性膝关节骨关节炎与超重、吸烟和激素治疗有关

Sandmark, H; Hogstedt, C; Lewold, S; Vingård, E