日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design of Bicyclic Peptide Tandems Mimicking the Homodimeric GDF15 Protein to Inhibit GDF15-GFRaL-RET Complex Cell Signaling

设计模拟同源二聚体GDF15蛋白的双环肽串联体以抑制GDF15-GFRaL-RET复合物细胞信号传导

Noisier, Anaïs F M; Sandmark, Jenny; Edfeldt, Fredrik; Backmark, Anna; Broddefalk, Johan; Wandzik, Joanna; Jurva, Ulrik; Ek, Margareta; Johansson, Carina A; Barlind, Louise; Gunnarsson, Jenny; Bigalke, Janna M; Xue, Yafeng; Frolov, Andrey I; Kankkonen, Cecilia; Roth, Robert G; Fritsch, Maria; Watcham, Sophie; van Rietschoten, Katerine; Mudd, Gemma E; Harrison, Helen; Chen, Liuhong; Skynner, Michael J; Craik, David J; Chankeshwara, Sunay V; Lemurell, Malin

Design of Selective sPLA(2)-X Inhibitor (-)-2-{2-[Carbamoyl-6-(trifluoromethoxy)-1H-indol-1-yl]pyridine-2-yl}propanoic Acid

选择性 sPLA(2)-X 抑制剂 (-)-2-{2-[氨基甲酰基-6-(三氟甲氧基)-1H-吲哚-1-基]吡啶-2-基}丙酸的设计

Giordanetto, Fabrizio; Knerr, Laurent; Nordberg, Peter; Pettersen, Daniel; Selmi, Nidhal; Beisel, Hans-Georg; de la Motte, Hannah; Månsson, Åsa; Dahlström, Mikael; Broddefalk, Johan; Saarinen, Gabrielle; Klingegård, Fredrik; Hurt-Camejo, Eva; Rosengren, Birgitta; Wikström, Johannes; Wågberg, Maria; Brengdahl, Johan; Rohman, Mattias; Sandmark, Jenny; Åkerud, Tomas; Roth, Robert G; Jansen, Frank; Ahlqvist, Marie

Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A(2) Type X (sPLA(2)-X) Inhibitors.

发现一系列吲哚-2 甲酰胺类化合物作为选择性分泌型磷脂酶 A(2) X 型 (sPLA(2)-X) 抑制剂

Knerr Laurent, Giordanetto Fabrizio, Nordberg Peter, Pettersen Daniel, Selmi Nidhal, Beisel Hans-Georg, de la Motte Hannah, Olsson Thomas, Perkins Tim D J, Herslöf Margareta, Månsson à sa, Dahlström Mikael, Starke Ingemar, Broddefalk Johan, Saarinen Gabrielle, Klingegård Fredrik, Hurt-Camejo Eva, Rosengren Birgitta, Brengdahl Johan, Jansen Frank, Rohman Mattias, Sandmark Jenny, Hallberg Kenth, à kerud Tomas, Roth Robert G, Ahlqvist Marie