日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Chemoproteomics validates selective targeting of Plasmodium M1 alanyl aminopeptidase as an antimalarial strategy

化学蛋白质组学验证了选择性靶向疟原虫 M1 丙氨酰氨基肽酶作为抗疟策略

Carlo Giannangelo #, Matthew P Challis #, Ghizal Siddiqui, Rebecca Edgar, Tess R Malcolm, Chaille T Webb, Nyssa Drinkwater, Natalie Vinh, Christopher Macraild, Natalie Counihan, Sandra Duffy, Sergio Wittlin, Shane M Devine, Vicky M Avery, Tania De Koning-Ward, Peter Scammells, Sheena McGowan, Darren

On-target, dual aminopeptidase inhibition provides cross-species antimalarial activity

靶向双氨基肽酶抑制提供跨物种抗疟活性

Rebecca C S Edgar, Tess R Malcolm, Ghizal Siddiqui, Carlo Giannangelo, Natalie A Counihan, Matthew Challis, Sandra Duffy, Mrittika Chowdhury, Jutta Marfurt, Madeline Dans, Grennady Wirjanata, Rintis Noviyanti, Kajal Daware, Chathura D Suraweera, Ric N Price, Sergio Wittlin, Vicky M Avery, Nyssa Drin

An adaptable, fit-for-purpose screening approach with high-throughput capability to determine speed of action and stage specificity of anti-malarial compounds

一种适应性强、适合用途的高通量筛选方法,用于确定抗疟化合物的作用速度和阶段特异性

Sandra Duffy, Brad E Sleebs, Vicky M Avery

Enhancing the Intrinsic Antiplasmodial Activity and Improving the Stability and Selectivity of a Tunable Peptide Scaffold Derived from Human Platelet Factor 4

增强内在抗疟原虫活性并提高源自人血小板因子 4 的可调肽支架的稳定性和选择性

Nicole Lawrence, Thomas N G Handley, Simon J de Veer, Maxim D Harding, Alicja Andraszek, Lachlan Hall, Karoline D Raven, Sandra Duffy, Vicky M Avery, David J Craik, Lara R Malins, Brendan J McMorran

Carbapenem-resistant Acinetobacter baumannii and Carbapenem-resistant Enterobacterales in US Dialysis Populations, 2016-2021

2016-2021年美国透析人群中耐碳青霉烯类鲍曼不动杆菌和耐碳青霉烯类肠杆菌科细菌的分布情况

Goff, Debra A; Du, Timothy; Baekyung Choi, Kelly; Silva, Anada; Lybeck, Cassandra; Golding, George; Hizon, Romeo; Ahmed, Sean; Chow, Blanda; Davis, Ian; Engbretson, Meghan; Evans, Gerald; Frenette, Charles; Johnstone, Jennie; Kibsey, Pamela; Katz, Kevin; Langley, Joanne; Leal, Jenine; Lee, Bonita; Longtin, Yves; Mertz, Dominik; Minion, Jessica; Science, Michelle; Srigley, Jocelyn; Suh, Kathryn; Titoria, Reena; Thampi, Nisha; Wong, Alice; Comeau, Jeannette; Hota, Susy; Gomes, Danica; Grass, Julian; Bulens, Sandra; Duffy, Nadezhda; Brandenburg, Joshua; Jacob, Jesse; Smith, Gillian; Vaeth, Elisabeth; Dumyati, Ghinwa; Flores, Kristina; Wilson, Christopher; Muleta, Daniel; Czaja, Christopher; Johnston, Helen; Lynfield, Ruth; Snippes Vagnone, Paula; O’Malley, Sean; Stabach, Nicole; Nadle, Joelle; Pierce, Rebecca; Guh, Alice; Novosad, Shannon; Cassidy, P Maureen

Synthesis and Antimalarial Evaluation of Halogenated Analogues of Thiaplakortone A

噻唑酮A卤代类似物的合成及抗疟活性评价

Folake A Egbewande, Brett D Schwartz, Sandra Duffy, Vicky M Avery, Rohan A Davis

Efficacy of Delafloxacin against the Biothreat Pathogen Burkholderia pseudomallei

德拉沙星对生物威胁病原体类鼻疽伯克霍尔德菌的疗效

McCurdy, Sandra; Duffy, Erin; Hickman, Mark; Halasohoris, Stephanie; Zumbrun, Steven D

Target Validation and Identification of Novel Boronate Inhibitors of the Plasmodium falciparum Proteasome

恶性疟原虫蛋白酶体新型硼酸盐抑制剂的靶标验证与鉴定

Stanley C Xie, David L Gillett, Natalie J Spillman, Christopher Tsu, Madeline R Luth, Sabine Ottilie, Sandra Duffy, Alexandra E Gould, Paul Hales, Benjamin A Seager, Carlie L Charron, Frank Bruzzese, Xiaofeng Yang, Xiansi Zhao, Shih-Chung Huang, Craig A Hutton, Jeremy N Burrows, Elizabeth A Winzeler

One-pot, multi-component synthesis and structure-activity relationships of peptoid-based histone deacetylase (HDAC) inhibitors targeting malaria parasites

针对疟原虫的基于肽的组蛋白去乙酰化酶 (HDAC) 抑制剂的一锅法多组分合成及构效关系

Daniela Diedrich, Katharina Stenzel, Eva Hesping, Yevgeniya Antonova-Koch, Tamirat Gebru, Sandra Duffy, Gillian Fisher, Andrea Schöler, Stephan Meister, Thomas Kurz, Vicky M Avery, Elizabeth A Winzeler, Jana Held, Katherine T Andrews, Finn K Hansen

Hexahydroquinolines are antimalarial candidates with potent blood-stage and transmission-blocking activity

六氢喹啉是具有强效血液阶段和传播阻断活性的抗疟药候选药物

Manu Vanaerschot, Leonardo Lucantoni, Tao Li, Jill M Combrinck, Andrea Ruecker, T R Santha Kumar, Kelly Rubiano, Pedro E Ferreira, Giulia Siciliano, Sonia Gulati, Philipp P Henrich, Caroline L Ng, James M Murithi, Victoria C Corey, Sandra Duffy, Ori J Lieberman, M Isabel Veiga, Robert E Sinden, Piet