日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cell membrane cholesterol affects serotonin transporter efflux due to altered transporter oligomerization

细胞膜胆固醇通过改变转运蛋白寡聚化影响血清素转运蛋白的外排。

Rudin, Deborah; Luethi, Dino; Niello, Marco; Yang, Jae-Won; Burger, Isabella; Sandtner, Walter; Birner-Gruenberger, Ruth; Schütz, Gerhard J; Sitte, Harald H

Revealing the location and dynamics of a concealed binding site in the dopamine transporter.

揭示多巴胺转运蛋白中隐藏结合位点的位置和动态

Zhu Rong, Sandtner Walter, Stockner Thomas, Heilinger Alexander, Holy Marion, Kudlacek Oliver, Wildling Linda, Saha Kusumika, Fröhlich Anna Sophie, Bindl Michael, Tziortzouda Paraskevi, Haider Anna, Gobl Julia, Suh Saanfor Hubert, Khan Jawad Akbar, Bicher Julia, Kastner Nina, Ebner Andreas, Gruber Hermann J, Freissmuth Michael, Newman Amy Hauck, Sitte Harald H, Hinterdorfer Peter

Careful Examination of a Novel Azobenzene Paroxetine Derivative and Its Interactions With Biogenic Amine Transporters.

仔细研究一种新型偶氮苯帕罗西汀衍生物及其与生物胺转运体的相互作用

Dreier Dominik, Belleza Oliver John V, Schlögl Katharina, Kickinger Stefanie, Hellsberg Eva, Mayer Felix P, Sandtner Walter, Mikšovsky Philipp, Schittmayer Matthias, Hu Yuntao, Jäntsch Kathrin, Holy Marion, Ecker Gerhard F, Sitte Harald H, Mihovilovic Marko D

Identification of the potassium-binding site in serotonin transporter

血清素转运蛋白中钾结合位点的鉴定

Hellsberg, Eva; Boytsov, Danila; Chen, Qingyang; Niello, Marco; Freissmuth, Michael; Rudnick, Gary; Zhang, Yuan-Wei; Sandtner, Walter; Forrest, Lucy R

Orphan lysosomal solute carrier MFSD1 facilitates highly selective dipeptide transport

孤儿溶酶体溶质载体 MFSD1 促进高度选择性二肽转运

Danila Boytsov, Gregor M Madej, Georg Horn, Nadine Blaha, Thomas Köcher, Harald H Sitte, Daria Siekhaus #, Christine Ziegler #, Walter Sandtner #, Marko Roblek

Structure-based discovery of conformationally selective inhibitors of the serotonin transporter

基于结构发现血清素转运蛋白的构象选择性抑制剂

Isha Singh, Anubha Seth, Christian B Billesbølle, Joao Braz, Ramona M Rodriguiz, Kasturi Roy, Bethlehem Bekele, Veronica Craik, Xi-Ping Huang, Danila Boytsov, Vladimir M Pogorelov, Parnian Lak, Henry O'Donnell, Walter Sandtner, John J Irwin, Bryan L Roth, Allan I Basbaum, William C Wetsel, Aashish M

Serotonin-releasing agents with reduced off-target effects

具有较低脱靶效应的血清素释放剂

Mayer, Felix P; Niello, Marco; Cintulova, Daniela; Sideromenos, Spyridon; Maier, Julian; Li, Yang; Bulling, Simon; Kudlacek, Oliver; Schicker, Klaus; Iwamoto, Hideki; Deng, Fei; Wan, Jinxia; Holy, Marion; Katamish, Rania; Sandtner, Walter; Li, Yulong; Pollak, Daniela D; Blakely, Randy D; Mihovilovic, Marko D; Baumann, Michael H; Sitte, Harald H

Persistent binding at dopamine transporters determines sustained psychostimulant effects

多巴胺转运蛋白上的持续结合决定了精神兴奋剂的持续作用

Niello, Marco; Sideromenos, Spyridon; Gradisch, Ralph; O Shea, Ronan; Schwazer, Jakob; Maier, Julian; Kastner, Nina; Sandtner, Walter; Jäntsch, Kathrin; Lupica, Carl R; Hoffman, Alexander F; Lubec, Gert; Loland, Claus J; Stockner, Thomas; Pollak, Daniela D; Baumann, Michael H; Sitte, Harald H

A mechanism of uncompetitive inhibition of the serotonin transporter

血清素转运蛋白的非竞争性抑制机制

Shreyas Bhat, Ali El-Kasaby, Ameya Kasture, Danila Boytsov, Julian B Reichelt, Thomas Hummel, Sonja Sucic, Christian Pifl, Michael Freissmuth, Walter Sandtner

Interactions of calmodulin kinase II with the dopamine transporter facilitate cocaine-induced enhancement of evoked dopamine release

钙调蛋白激酶II与多巴胺转运蛋白的相互作用促进可卡因诱导的多巴胺释放增强

Keighron, Jacqueline D; Bonaventura, Jordi; Li, Yang; Yang, Jae-Won; DeMarco, Emily M; Hersey, Melinda; Cao, Jianjing; Sandtner, Walter; Michaelides, Michael; Sitte, Harald H; Newman, Amy Hauck; Tanda, Gianluigi