日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

N-Boc-α-diazo glutarimide as efficient reagent for assembling N-heterocycle-glutarimide diads via Rh(II)-catalyzed N-H insertion reaction

N-Boc-α-重氮戊二酰亚胺作为高效试剂,可通过Rh(II)催化的NH插入反应组装N-杂环戊二酰亚胺二元体。

Kantin, Grigory; Golubev, Pavel; Sapegin, Alexander; Bunev, Alexander; Dar'in, Dmitry

Novel 5-Nitrofuran-Tagged Imidazo-Fused Azines and Azoles Amenable by the Groebke-Blackburn-Bienaymé Multicomponent Reaction: Activity Profile against ESKAPE Pathogens and Mycobacteria

新型5-硝基呋喃标记的咪唑稠合嗪和唑类化合物可通过Groebke-Blackburn-Bienaymé多组分反应合成:针对ESKAPE病原体和分枝杆菌的活性分析

Sapegin, Alexander; Rogacheva, Elizaveta; Kraeva, Lyudmila; Gureev, Maxim; Dogonadze, Marine; Vinogradova, Tatiana; Yablonsky, Petr; Balalaie, Saeed; Baykov, Sergey V; Krasavin, Mikhail

Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII

幸运的转变:咪唑啉类人碳酸酐酶VII抑制剂的效力和选择性显著提高

Kalinin, Stanislav; Kopylov, Stanislav; Tuccinardi, Tiziano; Sapegin, Alexander; Dar'in, Dmitry; Angeli, Andrea; Supuran, Claudiu T; Krasavin, Mikhail