日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The dual HCK/BTK inhibitor KIN-8194 impairs growth and integrin-mediated adhesion of BTKi-resistant mantle cell lymphoma

HCK/BTK 双重抑制剂 KIN-8194 可抑制 BTKi 耐药套细胞淋巴瘤的生长和整合素介导的粘附

Hildo C Lantermans, Fangxue Ma, Annemieke Kuil, Sanne van Kesteren, Sevtap Yasinoglu, Guang Yang, Sara J Buhrlage, Jinhua Wang, Nathanael S Gray, Marie José Kersten, Steven P Treon, Steven T Pals, Marcel Spaargaren

The dual HCK/BTK inhibitor KIN-8194 impairs growth and integrin-mediated adhesion of BTKi-resistant mantle cell lymphoma

双重 HCK/BTK 抑制剂 KIN-8194 可抑制 BTKi 耐药的套细胞淋巴瘤的生长和整合素介导的黏附。

Hildo C Lantermans ,Fangxue Ma ,Annemieke Kuil ,Sanne van Kesteren ,Sevtap Yasinoglu ,Guang Yang ,Sara J Buhrlage,Jinhua Wang,Nathanael S Gray,Marie José Kersten,Steven P Treon,Steven T Pals ,Marcel Spaargaren

Synergy between BRD9- and IKZF3-Targeting as a Therapeutic Strategy for Multiple Myeloma

BRD9 和 IKZF3 靶向协同作用作为多发性骨髓瘤治疗策略

Basudev Chowdhury, Swati Garg, Wei Ni, Martin Sattler, Dana Sanchez, Chengcheng Meng, Taisei Akatsu, Richard Stone, William Forrester, Edmund Harrington, Sara J Buhrlage, James D Griffin, Ellen Weisberg

Accelerating inhibitor discovery for deubiquitinating enzymes

加速发现去泛素化酶抑制剂

Wai Cheung Chan # ,Xiaoxi Liu # ,Robert S Magin ,Nicholas M Girardi ,Scott B Ficarro ,Wanyi Hu ,Maria I Tarazona Guzman ,Cara A Starnbach ,Alejandra Felix ,Guillaume Adelmant ,Anthony C Varca ,Bin Hu ,Ariana S Bratt ,Ethan DaSilva ,Nathan J Schauer ,Isabella Jaen Maisonet ,Emma K Dolen ,Anthony X Ayala ,Jarrod A Marto ,Sara J Buhrlage

KSHV Viral Protein Kinase Interacts with USP9X to Modulate the Viral Lifecycle

KSHV 病毒蛋白激酶与 USP9X 相互作用调节病毒生命周期

Danielle L Chappell, Praneet K Sandhu, Jason P Wong, Aadra P Bhatt, Xiaoxi Liu, Sara J Buhrlage, Brenda R S Temple, M Ben Major, Blossom Damania

Akkermansia muciniphila phospholipid induces homeostatic immune responses

Akkermansia muciniphila 磷脂诱导稳态免疫反应

Munhyung Bae #, Chelsi D Cassilly #, Xiaoxi Liu, Sung-Moo Park, Betsabeh Khoramian Tusi, Xiangjun Chen, Jaeyoung Kwon, Pavel Filipčík, Andrew S Bolze, Zehua Liu, Hera Vlamakis, Daniel B Graham, Sara J Buhrlage, Ramnik J Xavier, Jon Clardy

Akkermansia muciniphila phospholipid induces homeostatic immune responses

阿克曼氏菌磷脂诱导稳态免疫反应

Munhyung Bae #,Chelsi D Cassilly #,Xiaoxi Liu,Sung-Moo Park ,Betsabeh Khoramian Tusi ,Xiangjun Chen ,Jaeyoung Kwon,Pavel Filipčík,Andrew S Bolze,Zehua Liu,Hera Vlamakis,Daniel B Graham ,Sara J Buhrlage,Ramnik J Xavier ,Jon Clardy

Reversal of viral and epigenetic HLA class I repression in Merkel cell carcinoma

默克尔细胞癌中病毒和表观遗传HLA I类抑制的逆转

Patrick C Lee ,Susan Klaeger ,Phuong M Le ,Keegan Korthauer ,Jingwei Cheng ,Varsha Ananthapadmanabhan ,Thomas C Frost ,Jonathan D Stevens ,Alan Yl Wong ,J Bryan Iorgulescu ,Anna Y Tarren ,Vipheaviny A Chea ,Isabel P Carulli ,Camilla K Lemvigh ,Christina B Pedersen ,Ashley K Gartin ,Siranush Sarkizova ,Kyle T Wright ,Letitia W Li ,Jason Nomburg ,Shuqiang Li ,Teddy Huang ,Xiaoxi Liu ,Lucas Pomerance ,Laura M Doherty ,Annie M Apffel ,Luke J Wallace ,Suzanna Rachimi ,Kristen D Felt ,Jacquelyn O Wolff ,Elizabeth Witten ,Wandi Zhang ,Donna Neuberg ,William J Lane ,Guanglan Zhang ,Lars R Olsen ,Manisha Thakuria ,Scott J Rodig ,Karl R Clauser ,Gabriel J Starrett ,John G Doench ,Sara J Buhrlage ,Steven A Carr ,James A DeCaprio ,Catherine J Wu ,Derin B Keskin

Small molecule inhibition of deubiquitinating enzyme JOSD1 as a novel targeted therapy for leukemias with mutant JAK2

小分子抑制去泛素化酶 JOSD1 作为 JAK2 突变白血病的新型靶向疗法

Jing Yang #, Ellen L Weisberg #, Xiaoxi Liu #, Robert S Magin, Wai Cheung Chan, Bin Hu, Nathan J Schauer, Shengzhe Zhang, Ilaria Lamberto, Laura Doherty, Chengcheng Meng, Martin Sattler, Lucia Cabal-Hierro, Eric Winer, Richard Stone, Jarrod A Marto, James D Griffin, Sara J Buhrlage

Integrating multi-omics data reveals function and therapeutic potential of deubiquitinating enzymes

整合多组学数据揭示去泛素化酶的功能和治疗潜力

Laura M Doherty, Caitlin E Mills, Sarah A Boswell, Xiaoxi Liu, Charles Tapley Hoyt, Benjamin Gyori, Sara J Buhrlage, Peter K Sorger