日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of new 4-(6-oxopyridazin-1-yl)benzenesulfonamides as multi-target anti-inflammatory agents targeting carbonic anhydrase, COX-2 and 5-LOX enzymes: synthesis, biological evaluations and modelling insights

鉴定新的 4-(6-氧代吡嗪-1-基)苯磺酰胺作为针对碳酸酐酶、COX-2 和 5-LOX 酶的多靶点抗炎药物:合成、生物学评价和建模见解

Waleed A Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M Abd-Alhaseeb, Sara T Al-Rashood, Giri Babu Veerakanellore, Taghreed A Majrashi, Eslam B Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T Supuran, Wagdy M Eldehna, Mohamed Elagawany

Design and statistical optimisation of emulsomal nanoparticles for improved anti-SARS-CoV-2 activity of N-(5-nitrothiazol-2-yl)-carboxamido candidates: in vitro and in silico studies

乳化纳米粒子的设计和统计优化以提高 N-(5-硝基噻唑-2-基)-甲酰胺候选物的抗 SARS-CoV-2 活性:体外和计算机模拟研究

Ahmed A Al-Karmalawy, Dalia S El-Gamil, Rabeh El-Shesheny, Marwa Sharaky, Radwan Alnajjar, Omnia Kutkat, Yassmin Moatasim, Mohamed Elagawany, Sara T Al-Rashood, Faizah A Binjubair, Wagdy M Eldehna, Ayman M Noreddin, Mohamed Y Zakaria3

Synergistic Effect of Sophora japonica and Glycyrrhiza glabra Flavonoid-Rich Fractions on Wound Healing: In Vivo and Molecular Docking Studies

槐米和光果甘草富含黄酮类成分对伤口愈合的协同作用:体内和分子对接研究

Shaza H Aly, Ahmed M Elissawy, Abdulla M A Mahmoud, Fatma Sa'eed El-Tokhy, Sherif S Abdel Mageed, Hadia Almahli, Sara T Al-Rashood, Faizah A Binjubair, Mahmoud A El Hassab, Wagdy M Eldehna, Abd El-Nasser B Singab

Novel 3-(6-methylpyridin-2-yl)coumarin-based chalcones as selective inhibitors of cancer-related carbonic anhydrases IX and XII endowed with anti-proliferative activity

新型 3-(6-甲基吡啶-2-基)香豆素基查耳酮作为具有抗增殖活性的癌症相关碳酸酐酶 IX 和 XII 的选择性抑制剂

Haytham O Tawfik, Moataz A Shaldam, Alessio Nocentini, Rofaida Salem, Hadia Almahli, Sara T Al-Rashood, Claudiu T Supuran, Wagdy M Eldehna

Development of 2-oindolin-3-ylidene-indole-3-carbohydrazide derivatives as novel apoptotic and anti-proliferative agents towards colorectal cancer cells

2-吲哚-3-亚甲基吲哚-3-碳酰肼衍生物作为针对结直肠癌细胞的新型凋亡和抗增殖药物的开发

Wagdy M Eldehna, Mahmoud F Abo-Ashour, Tarfah Al-Warhi, Sara T Al-Rashood, Amal Alharbi, Rezk R Ayyad, Khayal Al-Khayal, Maha Abdulla, Hatem A Abdel-Aziz, Rehan Ahmad, Radwan El-Haggar

Synthesis and in vitro anticancer activity of certain novel 1-(2-methyl-6-arylpyridin-3-yl)-3-phenylureas as apoptosis-inducing agents

某些新型 1-(2-甲基-6-芳基吡啶-3-基)-3-苯基脲作为凋亡诱导剂的合成及体外抗癌活性

Wagdy M Eldehna, Ghada S Hassan, Sara T Al-Rashood, Tarfah Al-Warhi, Ahmed E Altyar, Hamad M Alkahtani, Abdulrahman A Almehizia, Hatem A Abdel-Aziz