日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-guided optimization of adenosine mimetics as selective and potent inhibitors of coronavirus nsp14 N7-methyltransferases

腺苷类似物的结构引导优化作为冠状病毒 nsp14 N7-甲基转移酶的选择性和有效抑制剂

Marcel Hausdorff, Adrien Delpal, Sarah Barelier, Laura Nicollet, Bruno Canard, Franck Touret, Agathe Colmant, Bruno Coutard, Jean-Jacques Vasseur, Etienne Decroly, Françoise Debart

Increasing chemical space coverage by combining empirical and computational fragment screens

通过结合经验和计算碎片筛选来增加化学空间覆盖率

Sarah Barelier, Oliv Eidam, Inbar Fish, Johan Hollander, Francis Figaroa, Ruta Nachane, John J Irwin, Brian K Shoichet, Gregg Siegal