Complexation of histone deacetylase inhibitor belinostat to Cu(II) prevents premature metabolic inactivation in vitro and demonstrates potent anti-cancer activity in vitro and ex vivo in colon cancer
组蛋白去乙酰化酶抑制剂贝利诺司他与 Cu(II) 的络合可防止体外过早代谢失活,并在体外和离体结肠癌中表现出强大的抗癌活性
期刊:Cellular Oncology
影响因子:
doi:10.1007/s13402-023-00882-x
Ellen Finnegan, Wei Ding, Ziga Ude, Sara Terer, Tadhg McGivern, Anna M Blümel, Grainne Kirwan, Xinxin Shao, Flavia Genua, Xiaofei Yin, Alexander Kel, Sarinj Fattah, Parvathi A Myer, Sally-Ann Cryan, Jochen H M Prehn, Darran P O'Connor, Lorraine Brennan, Gregory Yochum, Celine J Marmion #, Sudipto Da