日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Hybrid SAR Property Modeling of Novel Cholinesterase Inhibitors

新型胆碱酯酶抑制剂的合成及混合 SAR 特性建模

Jiri Kos, Violetta Kozik, Dominika Pindjakova, Timotej Jankech, Adam Smolinski, Sarka Stepankova, Jan Hosek, Michal Oravec, Josef Jampilek, Andrzej Bak

Novel Benzene-Based Carbamates for AChE/BChE Inhibition: Synthesis and Ligand/Structure-Oriented SAR Study

用于 AChE/BChE 抑制的新型苯基氨基甲酸酯:合成和配体/结构导向的 SAR 研究

Andrzej Bak, Violetta Kozik, Dariusz Kozakiewicz, Kamila Gajcy, Daniel Jan Strub, Aleksandra Swietlicka, Sarka Stepankova, Ales Imramovsky, Jaroslaw Polanski, Adam Smolinski, Josef Jampilek

Proline-Based Carbamates as Cholinesterase Inhibitors

脯氨酸基氨基甲酸酯作为胆碱酯酶抑制剂

Hana Pizova, Marketa Havelkova, Sarka Stepankova, Andrzej Bak, Tereza Kauerova, Violetta Kozik, Michal Oravec, Ales Imramovsky, Peter Kollar, Pavel Bobal, Josef Jampilek1

1,3-substituted imidazolidine-2,4,5-triones: synthesis and inhibition of cholinergic enzymes

1,3-取代咪唑烷-2,4,5-三酮:合成及对胆碱能酶的抑制

Vladimir Pejchal, Sarka Stepankova, Zdenka Padelkova, Ales Imramovsky, Josef Jampilek