Discovery of ERD-1233 as a Potent and Orally Efficacious Estrogen Receptor PROTAC Degrader for the Treatment of ER+ Human Breast Cancer
发现 ERD-1233 是一种强效且口服有效的雌激素受体 PROTAC 降解剂,可用于治疗 ER+ 人类乳腺癌
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c01521
Acharyya, Ranjan Kumar; Rej, Rohan Kalyan; Hu, Biao; Chen, Zhixiang; Wu, Dimin; Lu, Jianfeng; Metwally, Hoda; McEachern, Donna; Wang, Yu; Jiang, Wei; Bai, Longchuan; Tošović, Jelena; Gersch, Christina L; Xu, Guozhang; Zhang, Weihong; Wu, WenXue; Priestley, E Scott; Sui, Zhihua; Sarkari, Farzad; Wen, Bo; Sun, Duxin; Rae, James M; Wang, Shaomeng