Discovery of Selective and Orally Bioavailable Heterobifunctional Degraders of Cyclin-Dependent Kinase 2
发现选择性且口服生物利用度高的细胞周期蛋白依赖性激酶2异双功能降解剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c01160
Collier, Philip N; Zheng, Xiaozhang; Ford, Melissa; Weiss, Matthew; Chen, Dapeng; Li, Kunhua; Growney, Joseph D; Yang, Annan; Sathappa, Murugappan; Breitkopf, Susanne B; Enerson, Brad; Liang, Tong; Paul, Atanu; Sawant, Rupa; Su, Lijing; Aversa, Robert J; Howarth, Charles; Sharma, Kirti; Williams, Juliet; Kwiatkowski, Nicholas P