日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Selective and Orally Bioavailable Heterobifunctional Degraders of Cyclin-Dependent Kinase 2

发现选择性且口服生物利用度高的细胞周期蛋白依赖性激酶2异双功能降解剂

Collier, Philip N; Zheng, Xiaozhang; Ford, Melissa; Weiss, Matthew; Chen, Dapeng; Li, Kunhua; Growney, Joseph D; Yang, Annan; Sathappa, Murugappan; Breitkopf, Susanne B; Enerson, Brad; Liang, Tong; Paul, Atanu; Sawant, Rupa; Su, Lijing; Aversa, Robert J; Howarth, Charles; Sharma, Kirti; Williams, Juliet; Kwiatkowski, Nicholas P

Identification of small molecule inhibitors of PPM1D using an integrated drug discovery platform.

利用综合药物发现平台鉴定PPM1D小分子抑制剂

Shaw Subrata, Jiang Wei, Rush Jason, Dumont Nancy, Kim John, Singh Ritu, Skepner Adam, Khodier Carol, Raffier Cerise, Murphy Zachary, Yan Ni, Schluter Cameron, Yu Xiao, Szuchnicki Mateusz, Sathappa Murugappan, Kahn Josephine, Sperling Adam S, Wagner Florence, McKinney David C, Gould Alexandra E, Garvie Colin W, Miller Peter G