日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A tailored tetravalent peptide displays dual functions to inhibit amyloid β production and aggregation

一种定制的四价肽具有双重功能,可抑制β淀粉样蛋白的生成和聚集。

Waka Sato ,Miho Watanabe-Takahashi ,Takuya Murata ,Naoko Utsunomiya-Tate ,Jun Motoyama ,Masataka Anzai ,Seiko Ishihara ,Nanako Nishioka ,Hina Uchiyama ,Juri Togashi ,Saeka Nishihara ,Kiyoshi Kawasaki ,Takashi Saito ,Takaomi C Saido ,Satoru Funamoto ,Kiyotaka Nishikawa

Curcumin Derivative GT863 Inhibits Amyloid-Beta Production via Inhibition of Protein N-Glycosylation

姜黄素衍生物 GT863 通过抑制蛋白质 N-糖基化来抑制淀粉样β蛋白的产生

Yasuomi Urano, Mina Takahachi, Ryo Higashiura, Hitomi Fujiwara, Satoru Funamoto, So Imai, Eugene Futai, Michiaki Okuda, Hachiro Sugimoto, Noriko Noguchi

Affinity-Based Screening of Tetravalent Peptides Identifies Subtype-Selective Neutralizers of Shiga Toxin 2d, a Highly Virulent Subtype, by Targeting a Unique Amino Acid Involved in Its Receptor Recognition

基于亲和力的四价肽筛选通过靶向参与受体识别的独特氨基酸来鉴定志贺毒素 2d(一种高毒性亚型)的亚型选择性中和剂

Takaaki Mitsui, Miho Watanabe-Takahashi, Eiko Shimizu, Baihao Zhang, Satoru Funamoto, Shinji Yamasaki, Kiyotaka Nishikawa

Substrate ectodomain is critical for substrate preference and inhibition of γ-secretase

底物胞外域对于底物偏好和 γ-分泌酶抑制至关重要

Satoru Funamoto, Toru Sasaki, Seiko Ishihara, Mika Nobuhara, Masaki Nakano, Miho Watanabe-Takahashi, Takashi Saito, Nobuto Kakuda, Tomohiro Miyasaka, Kiyotaka Nishikawa, Takaomi C Saido, Yasuo Ihara

Modulation of lipid kinase PI4KIIα activity and lipid raft association of presenilin 1 underlies γ-secretase inhibition by ginsenoside (20S)-Rg3

人参皂苷 (20S)-Rg3 抑制 γ-分泌酶的基础是调节脂质激酶 PI4KIIα 活性和早老素 1 的脂筏结合

Min Suk Kang, Seung-Hoon Baek, Yoon Sun Chun, A Zenobia Moore, Natalie Landman, Diego Berman, Hyun Ok Yang, Maho Morishima-Kawashima, Satoko Osawa, Satoru Funamoto, Yasuo Ihara, Gilbert Di Paolo, Jeong Hill Park, Sungkwon Chung, Tae-Wan Kim

gamma-Secretase: successive tripeptide and tetrapeptide release from the transmembrane domain of beta-carboxyl terminal fragment

γ-分泌酶:从β-羧基末端片段的跨膜结构域连续释放三肽和四肽

Mako Takami, Yu Nagashima, Yoshihisa Sano, Seiko Ishihara, Maho Morishima-Kawashima, Satoru Funamoto, Yasuo Ihara