EPZ011989, A Potent, Orally-Available EZH2 Inhibitor with Robust in Vivo Activity
EPZ011989,一种高效、口服有效的EZH2抑制剂,具有显著的体内活性。
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5b00037
Campbell, John E; Kuntz, Kevin W; Knutson, Sarah K; Warholic, Natalie M; Keilhack, Heike; Wigle, Tim J; Raimondi, Alejandra; Klaus, Christine R; Rioux, Nathalie; Yokoi, Akira; Kawano, Satoshi; Minoshima, Yukinori; Choi, Hyeong-Wook; Porter Scott, Margaret; Waters, Nigel J; Smith, Jesse J; Chesworth, Richard; Moyer, Mikel P; Copeland, Robert A