Design of BET Inhibitor Bottlebrush Prodrugs with Superior Efficacy and Devoid of Systemic Toxicities
设计具有优异疗效且无全身毒性的BET抑制剂瓶刷状前药
期刊:Journal of the American Chemical Society
影响因子:15.6
doi:10.1021/jacs.1c00312
Vohidov, Farrukh; Andersen, Jannik N; Economides, Kyriakos D; Shipitsin, Michail V; Burenkova, Olga; Ackley, James C; Vangamudi, Bhavatarini; Nguyen, Hung V-T; Gallagher, Nolan M; Shieh, Peyton; Golder, Matthew R; Liu, Jenny; Dahlberg, William K; Ehrlich, Deborah J C; Kim, Julie; Kristufek, Samantha L; Huh, Sung Jin; Neenan, Allison M; Baddour, Joelle; Paramasivan, Sattanathan; de Stanchina, Elisa; Kc, Gaurab; Turnquist, David J; Saucier-Sawyer, Jennifer K; Kopesky, Paul W; Brady, Samantha W; Jessel, Michael J; Reiter, Lawrence A; Chickering, Donald E; Johnson, Jeremiah A; Blume-Jensen, Peter