Discovery of SY-5609: A Selective, Noncovalent Inhibitor of CDK7
SY-5609 的发现:一种选择性、非共价 CDK7 抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.1c01171
Jason J Marineau, Kristin B Hamman, Shanhu Hu, Sydney Alnemy, Janessa Mihalich, Anzhelika Kabro, Kenneth Matthew Whitmore, Dana K Winter, Stephanie Roy, Stephane Ciblat, Nan Ke, Anneli Savinainen, Ashraf Wilsily, Goran Malojcic, Robert Zahler, Darby Schmidt, Michael J Bradley, Nigel J Waters, Claudi