日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Inhibition of endocannabinoid hydrolases MAGL, FAAH and ABHD6 by AKU-005 reduces ex vivo cortical spreading depression

AKU-005 对内源性大麻素水解酶 MAGL、FAAH 和 ABHD6 的抑制可减少离体皮质扩散抑制

Brugia, Flavia; Ivanov, Konstantin; Aroviita, Auni; Giniatullina, Raisa; Lehtonen, Marko; Malm, Tarja; Savinainen, Juha; Giniatullin, Rashid; Della Pietra, Adriana

Correction: Inhibition of endocannabinoid hydrolases MAGL, FAAH and ABHD6 by AKU‑005 reduces ex vivo cortical spreading depression

更正:AKU-005 对内源性大麻素水解酶 MAGL、FAAH 和 ABHD6 的抑制作用可减轻离体皮质扩散性抑制

Brugia, Flavia; Ivanov, Konstantin; Aroviita, Auni; Giniatullina, Raisa; Lehtonen, Marko; Malm, Tarja; Savinainen, Juha; Giniatullin, Rashid; Pietra, Adriana Della

Differential inhibitory effects of endocannabinoids on neuronal firing of mouse meningeal afferents

内源性大麻素对小鼠脑膜传入神经元放电的差异性抑制作用

Krivoshein, Georgii; Della Pietra, Adriana; Savinainen, Juha; van den Maagdenberg, Arn M J M; Giniatullin, Rashid

Synovial fluid o-tyrosine is a potential biomarker for autoimmune-driven rheumatoid arthritis

滑液中邻酪氨酸是自身免疫性类风湿性关节炎的潜在生物标志物

Mustonen, Anne-Mari; Savinainen, Juha; Lehtonen, Marko; Lehenkari, Petri; Kääriäinen, Tommi; Joukainen, Antti; Kröger, Heikki; Nieminen, Petteri

5-Aminothiazoles Reveal a New Ligand-Binding Site on Prolyl Oligopeptidase Which is Important for Modulation of Its Protein-Protein Interaction-Derived Functions

5-氨基噻唑揭示了脯氨酰寡肽酶上的新配体结合位点,这对调节其蛋白质-蛋白质相互作用衍生的功能很重要

Henri T Pätsi, Tommi P Kilpeläinen, Mikael Jumppanen, Johanna Uhari-Väänänen, Pieter Van Wielendaele, Francesca De Lorenzo, Hengjing Cui, Samuli Auno, Janne Saharinen, Erin Seppälä, Nina Sipari, Juha Savinainen, Ingrid De Meester, Anne-Marie Lambeir, Maija Lahtela-Kakkonen, Timo T Myöhänen, Erik A A

Social and health care top managers' perceptions and aims of strategic work ability management in the midst of change

社会和医疗保健高层管理者在变革中对战略性工作能力管理的认知和目标

Anttilainen, Julia; Pehkonen, Irmeli; Savinainen, Minna; Haukka, Eija

Immune checkpoint inhibition combined with targeted therapy using a novel virus-like drug conjugate induces complete responses in a murine model of local and distant tumors

免疫检查点抑制与使用新型病毒样药物偶联物的靶向治疗相结合,可在小鼠局部和远处肿瘤模型中诱导完全缓解

Ruben V Huis In 't Veld, Sen Ma, Rhonda C Kines, Anneli Savinainen, Cadmus Rich, Ferry Ossendorp, Martine J Jager

Potent dual MAGL/FAAH inhibitor AKU-005 engages endocannabinoids to diminish meningeal nociception implicated in migraine pain

强效双重 MAGL/FAAH 抑制剂 AKU-005 与内源性大麻素结合,减轻与偏头痛有关的脑膜痛

Adriana Della Pietra #, Georgii Krivoshein #, Konstantin Ivanov, Raisa Giniatullina, Henna-Kaisa Jyrkkänen, Ville Leinonen, Marko Lehtonen, Arn M J M van den Maagdenberg, Juha Savinainen, Rashid Giniatullin

Discovery of SY-5609: A Selective, Noncovalent Inhibitor of CDK7

SY-5609 的发现:一种选择性、非共价 CDK7 抑制剂

Jason J Marineau, Kristin B Hamman, Shanhu Hu, Sydney Alnemy, Janessa Mihalich, Anzhelika Kabro, Kenneth Matthew Whitmore, Dana K Winter, Stephanie Roy, Stephane Ciblat, Nan Ke, Anneli Savinainen, Ashraf Wilsily, Goran Malojcic, Robert Zahler, Darby Schmidt, Michael J Bradley, Nigel J Waters, Claudi

Determinants of Cognitive Performance in Children and Adolescents: A Populational Longitudinal Study

儿童和青少年认知能力的决定因素:一项人口纵向研究

Lima, Rodrigo Antunes; Soares, Fernanda Cunha; van Poppel, Mireille; Savinainen, Saija; Mäntyselkä, Aino; Haapala, Eero A; Lakka, Timo