Discovery of the SARS-CoV-2 Papain-Like Protease Inhibitor MR1-114: From Structure-Based Design to In Vivo Antiviral Efficacy
SARS-CoV-2木瓜蛋白酶样蛋白酶抑制剂MR1-114的发现:从基于结构的药物设计到体内抗病毒功效
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c03846
Gannarapu, Malla Reddy; Indukuri, Divakar; Holberg, Cameron; Ratia, Kiira; Ramos, Omar Lozano; Cardoza, Savio; Velma, Ganga Reddy; Musku, Soumya Reddy; Qi, Zuohuang; Slilaty, Steve; Li, Zuomei; Rong, Lijun; Thatcher, Gregory R J; Xiong, Rui