日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Overcoming Ligand Discovery Challenges: Developing Peptide-Based Tracers for SPSB2

克服配体发现挑战:开发用于 SPSB2 的基于肽的示踪剂

Lenz, Christopher; Elson, Lewis; Dopfer, Johannes; Farges, Frederic; Krämer, Andreas; Löhr, Frank; Müller, Susanne; Guéret, Stéphanie M; Waldmann, Herbert; Dötsch, Volker; Saxena, Krishna; Knapp, Stefan

Biochemical investigation of LC3/GABARAP-ligand interaction as an important quality measure for LC3/GABARAP-targeting small molecules: addendum to the guidelines (4th edition)

LC3/GABARAP-配体相互作用的生化研究作为LC3/GABARAP靶向小分子药物的重要质量指标:指南补充(第四版)

Schwalm, Martin P; Lenz, Christopher; Saxena, Krishna; Klionsky, Daniel J; Proschak, Ewgenij; Knapp, Stefan

Crystallographic fragment screening reveals ligand hotspots in TRIM21 PRY-SPRY domain.

晶体学片段筛选揭示了TRIM21 PRY-SPRY结构域中的配体热点

Kim Yeojin, Lučić Aleksandar, Lenz Christopher, Farges Frederic, Schwalm Martin P, Saxena Krishna, Hanke Thomas, Marples Peter G, Aschenbrenner Jasmin C, Fearon Daren, von Delft Frank, Krämer Andreas, Knapp Stefan

Un-LOK-ing a New Approach for Conformational Selective Targeting of STK10 (LOK)

针对 STK10 (LOK) 构象选择性靶向的新方法——解构 LOK

Dettenhöfer, Martina; Tandara, Laura Nadine; Amrhein, Jennifer Alisa; Kurz, Christian Georg; Schwalm, Martin Peter; Mensing, Theresa Elisabeth; Wahl, Laurenz Maximilian; Krämer, Andreas; Gerninghaus, Joshua; Lenz, Christopher; Elson, Lewis; Berger, Benedict-Tilman; Schröder, Martin; Saxena, Krishna; Müller, Susanne; Knapp, Stefan; Greco, Francesco Aleksy; Hanke, Thomas

Back-Pocket Optimization of 2-Aminopyrimidine-Based Macrocycles Leads to Potent EPHA2/GAK Kinase Inhibitors.

2-氨基嘧啶基大环化合物的后口袋优化可得到强效的EPHA2/GAK激酶抑制剂

Gerninghaus Joshua, Zhubi Rezart, Krämer Andreas, Karim Marwah, Tran Do Hoang Nhu, Joerger Andreas C, Schreiber Christian, Berger Lena M, Berger Benedict-Tilman, Ehret Theresa A L, Elson Lewis, Lenz Christopher, Saxena Krishna, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas

NMR resonance assignment of a fibroblast growth factor 8 splicing isoform b

成纤维细胞生长因子 8 剪接异构体 b 的 NMR 共振归属

Hargittay, Bruno; Mineev, Konstantin S; Richter, Christian; Sreeramulu, Sridhar; Jonker, Hendrik R A; Saxena, Krishna; Schwalbe, Harald

Correction to 'Secondary structure determination of conserved SARS-CoV-2 RNA elements by NMR spectroscopy'

对“利用核磁共振波谱法测定SARS-CoV-2 RNA保守元件的二级结构”一文的更正

Wacker, Anna; Weigand, Julia E; Akabayov, Sabine R; Altincekic, Nadide; Bains, Jasleen Kaur; Banijamali, Elnaz; Binas, Oliver; Castillo-Martinez, Jesus; Cetiner, Erhan; Ceylan, Betül; Chiu, Liang-Yuan; Davila-Calderon, Jesse; Dhamotharan, Karthikeyan; Duchardt-Ferner, Elke; Ferner, Jan; Frydman, Lucio; Fürtig, Boris; Gallego, José; Grün, J Tassilo; Hacker, Carolin; Haddad, Christina; Hähnke, Martin; Hengesbach, Martin; Hiller, Fabian; Hohmann, Katharina F; Hymon, Daniel; de Jesus, Vanessa; Jonker, Henry; Keller, Heiko; Knezic, Bozana; Landgraf, Tom; Löhr, Frank; Luo, Le; Mertinkus, Klara R; Muhs, Christina; Novakovic, Mihajlo; Oxenfarth, Andreas; Palomino-Schätzlein, Martina; Petzold, Katja; Peter, Stephen A; Pyper, Dennis J; Qureshi, Nusrat S; Riad, Magdalena; Richter, Christian; Saxena, Krishna; Schamber, Tatjana; Scherf, Tali; Schlagnitweit, Judith; Schlundt, Andreas; Schnieders, Robbin; Schwalbe, Harald; Simba-Lahuasi, Alvaro; Sreeramulu, Sridhar; Stirnal, Elke; Sudakov, Alexey; Tants, Jan-Niklas; Tolbert, Blanton S; Vögele, Jennifer; Weiß, Lena; Wirmer-Bartoschek, Julia; Wirtz Martin, Maria A; Wöhnert, Jens; Zetzsche, Heidi

Large-Scale Recombinant Production of the SARS-CoV-2 Proteome for High-Throughput and Structural Biology Applications

用于高通量和结构生物学应用的SARS-CoV-2蛋白质组的大规模重组生产

Altincekic, Nadide; Korn, Sophie Marianne; Qureshi, Nusrat Shahin; Dujardin, Marie; Ninot-Pedrosa, Martí; Abele, Rupert; Abi Saad, Marie Jose; Alfano, Caterina; Almeida, Fabio C L; Alshamleh, Islam; de Amorim, Gisele Cardoso; Anderson, Thomas K; Anobom, Cristiane D; Anorma, Chelsea; Bains, Jasleen Kaur; Bax, Adriaan; Blackledge, Martin; Blechar, Julius; Böckmann, Anja; Brigandat, Louis; Bula, Anna; Bütikofer, Matthias; Camacho-Zarco, Aldo R; Carlomagno, Teresa; Caruso, Icaro Putinhon; Ceylan, Betül; Chaikuad, Apirat; Chu, Feixia; Cole, Laura; Crosby, Marquise G; de Jesus, Vanessa; Dhamotharan, Karthikeyan; Felli, Isabella C; Ferner, Jan; Fleischmann, Yanick; Fogeron, Marie-Laure; Fourkiotis, Nikolaos K; Fuks, Christin; Fürtig, Boris; Gallo, Angelo; Gande, Santosh L; Gerez, Juan Atilio; Ghosh, Dhiman; Gomes-Neto, Francisco; Gorbatyuk, Oksana; Guseva, Serafima; Hacker, Carolin; Häfner, Sabine; Hao, Bing; Hargittay, Bruno; Henzler-Wildman, K; Hoch, Jeffrey C; Hohmann, Katharina F; Hutchison, Marie T; Jaudzems, Kristaps; Jović, Katarina; Kaderli, Janina; Kalniņš, Gints; Kaņepe, Iveta; Kirchdoerfer, Robert N; Kirkpatrick, John; Knapp, Stefan; Krishnathas, Robin; Kutz, Felicitas; Zur Lage, Susanne; Lambertz, Roderick; Lang, Andras; Laurents, Douglas; Lecoq, Lauriane; Linhard, Verena; Löhr, Frank; Malki, Anas; Bessa, Luiza Mamigonian; Martin, Rachel W; Matzel, Tobias; Maurin, Damien; McNutt, Seth W; Mebus-Antunes, Nathane Cunha; Meier, Beat H; Meiser, Nathalie; Mompeán, Miguel; Monaca, Elisa; Montserret, Roland; Mariño Perez, Laura; Moser, Celine; Muhle-Goll, Claudia; Neves-Martins, Thais Cristtina; Ni, Xiamonin; Norton-Baker, Brenna; Pierattelli, Roberta; Pontoriero, Letizia; Pustovalova, Yulia; Ohlenschläger, Oliver; Orts, Julien; Da Poian, Andrea T; Pyper, Dennis J; Richter, Christian; Riek, Roland; Rienstra, Chad M; Robertson, Angus; Pinheiro, Anderson S; Sabbatella, Raffaele; Salvi, Nicola; Saxena, Krishna; Schulte, Linda; Schiavina, Marco; Schwalbe, Harald; Silber, Mara; Almeida, Marcius da Silva; Sprague-Piercy, Marc A; Spyroulias, Georgios A; Sreeramulu, Sridhar; Tants, Jan-Niklas; Tārs, Kaspars; Torres, Felix; Töws, Sabrina; Treviño, Miguel Á; Trucks, Sven; Tsika, Aikaterini C; Varga, Krisztina; Wang, Ying; Weber, Marco E; Weigand, Julia E; Wiedemann, Christoph; Wirmer-Bartoschek, Julia; Wirtz Martin, Maria Alexandra; Zehnder, Johannes; Hengesbach, Martin; Schlundt, Andreas

NMR Spectroscopic Characterization of the C-Mannose Conformation in a Thrombospondin Repeat Using a Selective Labeling Approach

利用选择性标记方法对血小板反应蛋白重复序列中的C-甘露糖构象进行核磁共振波谱表征

Jonker, Hendrik R A; Saxena, Krishna; Shcherbakova, Aleksandra; Tiemann, Birgit; Bakker, Hans; Schwalbe, Harald

Light Dynamics of the Retinal-Disease-Relevant G90D Bovine Rhodopsin Mutant

与视网膜疾病相关的G90D牛视紫红质突变体的光动力学

Kubatova, Nina; Mao, Jiafei; Eckert, Carl Elias; Saxena, Krishna; Gande, Santosh L; Wachtveitl, Josef; Glaubitz, Clemens; Schwalbe, Harald