The Selective Estrogen Receptor Degrader ZN-c5 Has Broad Antitumor Activity in Wild-Type and Mutant ER-Positive Breast Cancer Models.
选择性雌激素受体降解剂 ZN-c5 在野生型和突变型 ER 阳性乳腺癌模型中具有广泛的抗肿瘤活性。
期刊:Molecular Cancer Therapeutics
影响因子:5.5
doi:10.1158/1535-7163.MCT-25-0315
Ma Jianhui, Hegde Sayee, Sergeeva Masha, Chakraborty Binita, Wardell Suzanne E, McDonnell Donald P, Huang Peter Q, Bunker Kevin D, Doñate Fernando, Lackner Mark R, Samatar Ahmed A