日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a potent anti-Zika virus benzamide series targeting the viral protein NS4B

发现一系列靶向病毒蛋白NS4B的强效抗寨卡病毒苯甲酰胺类化合物

Chung, Donghoon; Otsuka, Yuka; Kim, Eunjung; Ullah, Sultan; Kennedy, Nicole M; Ngo, Khac Huy; Kang, Jinjoo; Tomlinson, Reece; Alejandro, Brian; Barnaby, Koji; Miller, Jeffrey; Shumate, Justin; Teo, Chwee Fang; Tan, Yaw Bia; Chew, Che Shin; Kang, CongBao; Luo, Dahai; Scampavia, Louis; Spicer, Timothy P; Bannister, Thomas D

Selective Glucocorticoid Receptor Modulators of Immune Checkpoint Function

免疫检查点功能的选择性糖皮质激素受体调节剂

Kobylski, Robin R; Min, Charles K; Nwachukwu, Jerome C; Koenig, Marcel; Zhang, Haotian; Moncada, Lizbeth; Venables, Thomas T; Schell, Bin-Bin; Stein, William J; McCown, Claudia; Schumate, Justin; Bonilla, Emelie; Sobh, Amin; Romero-Toledo, Arantxa; Pipkin, Matthew E; Janiszewska, Michalina; Scampavia, Louis; Spicer, Timothy P; Licht, Jonathan D; Rogatsky, Inez; Kamenecka, Theodore M; Solt, Laura A; Nettles, Kendall W

Homeostatic scaling of dynorphin signaling by a non-canonical opioid receptor

非经典阿片受体介导的强啡肽信号稳态调节

Li, Xiaona; Winters, Nathan D; Pandey, Shubhi; Lankford, Colten; Stoveken, Hannah M; Smith, Emery; Chang, Chu-Ting; Zucca, Stefano; Scampavia, Louis; Spicer, Timothy; Martemyanov, Kirill A

The Endo-GeneScreen platform identifies drug-like probes that regulate endogenous protein levels within physiological contexts

Endo-GeneScreen平台能够识别在生理环境下调节内源性蛋白质水平的类药物探针。

Samowitz, Preston; Radnai, Laszlo; Vaissiere, Thomas; Michaelson, Sheldon D; Rojas, Camilo; Mitchell, Ryan; Kilinc, Murat; Edwards, Austin; Shumate, Justin; Hawkins, Richard; Fernandez-Vega, Virneliz; Spicer, Timothy P; Scampavia, Louis; Kamenecka, Theodore; Miller, Courtney A; Rumbaugh, Gavin

A high throughput assay for phosphoribosylformylglycinamidine synthase

磷酸核糖甲酰甘氨酰胺合酶的高通量检测方法

Sharma, Nandini; Otsuka, Yuka; Scampavia, Louis; Spicer, Timothy P; French, Jarrod B

Hyperphosphorylated tau-based Alzheimer's Disease drug discovery: Identification of inhibitors of tau aggregation and cytotoxicity.

基于过度磷酸化 tau 的阿尔茨海默病药物发现:tau 聚集和细胞毒性抑制剂的鉴定

Hagar Hsiao-Tien, Fernandez-Vega Virneliz, Wang Kuang-Wei, Jordan Luis M Ortiz, Shumate Justin, Scampavia Louis, Tapayan April Sweet, Nguyen Hien M, Spicer Timothy P, Kuo Min-Hao

Discovery of a potent anti-Zika virus benzamide series targeting the viral protein NS4B

发现一系列靶向病毒蛋白NS4B的强效抗寨卡病毒苯甲酰胺类化合物

Chung, Donghoon; Otsuka, Yuka; Kim, Eunjung; Ullah, Sultan; Kennedy, Nicole M; Ngo, Khac Huy; Kang, Jinjoo; Tomlison, Reece; Alejandro, Brian; Barnaby, Koji; Miller, Jeffery; Shumate, Justin; Teo, Chwee Fang; Tan, Yaw Bia; Chew, Che Shin; Kang, CongBao; Luo, Dahai; Scampavia, Louis; Spicer, Timothy P; Bannister, Thomas D

A SARS-CoV-2 entry inhibitor trimerizes to lock the spike protein in a closed conformation

SARS-CoV-2病毒入侵抑制剂三聚化,将刺突蛋白锁定在封闭构象中。

Mou, Huihui; Gao, Bo; Ye, Gang; Zhang, Lizhou; Saxena, Divyasha; Bu, Fan; Vishwakarma, Jyoti; Zhou, Shuo; Bayona, Claudia Ruiz; Lin, Li; Getmanenko, Yulia; Bhandari, Janarjan; Bailey, Charles C; Crynen, Gogce C; Kitzmiller, Claire E; Li, Hao; Otsuka, Yuka; Wang, Chao; Batra, Lalit; Weston, Stuart; Frieman, Matthew B; Meyerholz, David K; Scampavia, Louis; Spicer, Timothy P; Harris, Reuben S; Cameron, Michael D; Bannister, Thomas D; Zheng, Jian; Farzan, Michael; Li, Fang; Choe, Hyeryun

Target-based discovery of a broad-spectrum flukicide.

基于靶点的广谱杀吸虫剂的发现

Sprague Daniel J, Park Sang-Kyu, Gramberg Svenja, Bauer Lisa, Rohr Claudia M, Chulkov Evgeny G, Smith Emery, Scampavia Louis, Spicer Timothy P, Haeberlein Simone, Marchant Jonathan S

High throughput screening for SARS-CoV-2 helicase inhibitors

SARS-CoV-2解旋酶抑制剂的高通量筛选

Otsuka, Yuka; Kim, Eunjung; Krueger, Austin; Shumate, Justin; Wang, Chao; Bdiri, Bilel; Ullah, Sultan; Park, HaJeung; Scampavia, Louis; Bannister, Thomas D; Chung, Donghoon; Spicer, Timothy P