Discovery of the First Efficacious Adenosine 2A Receptor Negative Allosteric Modulators for High Adenosine Cancer Immunotherapies
发现首个高效的腺苷2A受体负变构调节剂用于高腺苷癌症免疫疗法
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c01691
Boujut, Margot; Héritier, Margaux; Gouiller, Aurélie; Süess, Camille; Scapozza, Alessandro; De Smedt, Thibaut; Guibert, Maxime; Tardy, Sébastien; Ismail, Hesham M; Pejoski, David; Scapozza, Leonardo