日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Host-directed treatments for tuberculous meningitis: A multi-platform approach across mouse and human models

针对结核性脑膜炎的宿主导向治疗:跨小鼠和人类模型的多平台方法

Jain, Sanjay; Gonzalez, Carlos Ruiz; Singh, Medha; Leon, Yuderleys Masias; Chen, Xueyi; Sarhan, Mona; Martinez-Martinez, Yazmin; Patel, Shruti; Shambles, Madelynn; Villabona-Rueda, Andres; Lissit, Kadia; Tweedie, David; Scerba, Michael; Bishai, William; Artemov, Dmitri; Xu, Jinchong; D'Alessio, Franco; Hafner, Richard; Greig, Nigel; Manion, Maura; Sereti, Irini

Correction: Batsaikhan et al. Post-Injury Neuroprotective Effects of the Thalidomide Analog 3,6'-Dithiothalidomide on Traumatic Brain Injury. Int. J. Mol. Sci. 2019, 20, 502

更正:Batsaikhan 等人,《沙利度胺类似物 3,6'-二硫代沙利度胺对创伤性脑损伤的损伤后神经保护作用》,《国际分子科学杂志》,2019 年,第 20 卷,第 502 页。

Batsaikhan, Buyandelger; Wang, Jing-Ya; Scerba, Michael T; Tweedie, David; Greig, Nigel H; Miller, Jonathan P; Hoffer, Barry J; Lin, Chih-Tung; Wang, Jia-Yi

2-(Piperidin-3-yl)phthalimides reduce classical markers of cellular inflammation in LPS-challenged RAW 264.7 cells and also demonstrate potentially relevant sigma and serotonin receptor affinity in membrane preparations

2-(哌啶-3-基)邻苯二甲酰亚胺可降低LPS刺激的RAW 264.7细胞中经典的细胞炎症标志物,并且在膜制备物中也表现出潜在的相关σ受体和血清素受体亲和力。

Scerba, Michael T; Tweedie, David; Greig, Nigel H

Repurposing Pomalidomide as a Neuroprotective Drug: Efficacy in an Alpha-Synuclein-Based Model of Parkinson's Disease

将泊马度胺重新定位为神经保护药物:在基于α-突触核蛋白的帕金森病模型中的疗效

Palmas, Maria Francesca; Ena, Anna; Burgaletto, Chiara; Casu, Maria Antonietta; Cantarella, Giuseppina; Carboni, Ezio; Etzi, Michela; De Simone, Alfonso; Fusco, Giuliana; Cardia, Maria Cristina; Lai, Francesco; Picci, Luca; Tweedie, David; Scerba, Michael T; Coroneo, Valentina; Bernardini, Renato; Greig, Nigel H; Pisanu, Augusta; Carta, Anna R

3,6'- and 1,6'-Dithiopomalidomide Mitigate Ischemic Stroke in Rats and Blunt Inflammation

3,6'-和1,6'-二硫代马来酸可减轻大鼠缺血性中风并抑制炎症

Yan-Rou Tsai ,Dong Seok Kim ,Shih-Chang Hsueh ,Kai-Yun Chen ,John Chung-Che Wu ,Jia-Yi Wang ,Yi-Syue Tsou ,Inho Hwang ,Yukyung Kim ,Dayeon Gil ,Eui Jung Jo ,Baek-Soo Han ,David Tweedie ,Daniela Lecca ,Michael T Scerba ,Warren R Selman ,Barry J Hoffer ,Nigel H Greig ,Yung-Hsiao Chiang

Activity of a Novel Anti-Inflammatory Agent F-3,6'-dithiopomalidomide as a Treatment for Traumatic Brain Injury

新型抗炎药F-3,6'-二硫代马来酸胺治疗创伤性脑损伤的活性

Shih Chang Hsueh ,Michael T Scerba ,David Tweedie ,Daniela Lecca ,Dong Seok Kim ,Abdul Mannan Baig ,Yu Kyung Kim ,Inho Hwang ,Sun Kim ,Warren R Selman ,Barry J Hoffer ,Nigel H Greig

Thionated aminofluorophthalimides reduce classical markers of cellular inflammation in LPS-challenged RAW 264.7 cells

硫代氨基氟邻苯二甲酰亚胺可降低LPS刺激的RAW 264.7细胞中经典的细胞炎症标志物。

Scerba, Michael T; Tweedie, David; Lecca, Daniela; Siegler, Maxime A; Rais, Rana; Greig, Nigel H

Repurposing Immunomodulatory Imide Drugs (IMiDs) in Neuropsychiatric and Neurodegenerative Disorders

免疫调节酰亚胺类药物(IMiDs)在神经精神疾病和神经退行性疾病中的再利用

Jung, Yoo Jin; Tweedie, David; Scerba, Michael T; Kim, Dong Seok; Palmas, Maria Francesca; Pisanu, Augusta; Carta, Anna R; Greig, Nigel H

3,6'-dithiopomalidomide reduces neural loss, inflammation, behavioral deficits in brain injury and microglial activation

3,6'-二硫代泊马度胺可减少脑损伤中的神经损失、炎症、行为缺陷以及小胶质细胞活化

Chih-Tung Lin #, Daniela Lecca #, Ling-Yu Yang #, Weiming Luo #, Michael T Scerba, David Tweedie, Pen-Sen Huang, Yoo-Jin Jung, Dong Seok Kim, Chih-Hao Yang, Barry J Hoffer, Jia-Yi Wang, Nigel H Greig

The structure-activity profile of mercaptobenzamides' anti-HIV activity suggests that thermodynamics of metabolism is more important than binding affinity to the target

巯基苯甲酰胺抗 HIV 活性的结构-活性特征表明,代谢热力学比与靶标的结合亲和力更重要

Herman Nikolayevskiy, Marco Robello, Michael T Scerba, Evan H Pasternak, Mrinmoy Saha, Tracy L Hartman, Caitlin A Buchholz, Robert W Buckheit Jr, Stewart R Durell, Daniel H Appella