日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An allele-agnostic mutant-KRAS inhibitor suppresses tumor maintenance signals and reprograms tumor immunity in pancreatic cancer

一种不依赖于特定等位基因的突变型KRAS抑制剂可抑制肿瘤维持信号并重编程胰腺癌的肿瘤免疫。

McAndrews, Kathleen M; Paradiso, Francesca; Stalnecker, Clint A; Chellakkan, Benson S; Thege, Fredrik I; Peng, David H; Moreno Diaz, Barbara A; Sugimoto, Hikaru; Patel, Sarah I; Mahadevan, Krishnan K; Kirtley, Michelle L; Wills, Danielle; Sockwell, Amari M; Fonseca, Andre Luis F; Liu, Yunhe; Rajapakshe, Kimal I; Yee, Nathaniel G; Tran, Phuong Thao; Omar, Huda Alchikh; Tedeschi, Antonio; Schischlik-Siegl, Fiorella; Boghossian, Andrew S; Rees, Matthew G; Ronan, Melissa M; Roth, Jennifer A; Rudolph, Dorothea; Aichinger, Martin; Ebner, Florian; Artemov, Artem V; Lipp, Jesse; Pisarsky, Laura; Herrmann, Valerie Laura; Park, John; Rippmann, Jörg F; Schaaf, Otmar; Chandler, Vanessa; Williams, Mariah; Deckard, Charles E; Wang, Linghua; Der, Channing J; Vellano, Christopher; Guerrero, Paola A; Heffernan, Timothy P; Kalluri, Raghu; Maitra, Anirban

Discovery of BI-2493, a Pan-KRAS Inhibitor Showing In Vivo Efficacy.

发现 BI-2493,一种泛 KRAS 抑制剂,显示出体内疗效

Bröker Joachim, Waterson Alex G, Hodges Timothy R, Abbott Jason R, Arnold Allison, Böttcher Jark, Braun Nina, Cui Jianwen, Fuchs Julian E, Gerstberger Thomas, Gogg Sebastian, Hanner Sabine, Herdeis Lorenz, Howell Lucas W, Mantoulidis Andreas, Mayer Moriz, Phan Jason, Rocchetti Francesca, Sankar Kyra, Sarkar Dhruba, Schaaf Otmar, Sensintaffar John L, Sun Qi, Wunberg Tobias, Fesik Stephen W