日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Saskemycin, a potent and selective antimycobacterial agent targeting a unique site on the ribosome.

Saskemycin 是一种强效且选择性的抗分枝杆菌药物,靶向核糖体上的独特位点。

Wright Gerard, Cook Michael, Xu Min, Morici Martino, Travin Dmitrii, Wang Wenliang, Klepacki Dorota, Chhabra Nandini, Rao Vishwas, Sahile Henok, Hackenberger Dirk, Safdari Haaris, Berger Max, Corazza Martina, Bond Austin, Guitor Allison, Tertigas Dominique, Wang Lijun, Schaenzer Adam, Ejim Linda, Yarlagadda Venkateswarlu, Gomez James, Surette Michael, Av-Gay Yossef, Dhar Neeraj, Hung Deborah, Vázquez-Laslop Nora, Mankin Alexander, Wilson Daniel

Identification and characterization of the siderochelin biosynthetic gene cluster via coculture

通过共培养鉴定和表征铁螯合素生物合成基因簇

Schaenzer, Adam J; Wang, Wenliang; Hackenberger, Dirk; Wright, Gerard D

Bacillus subtilis-derived peptides disrupt quorum sensing and biofilm assembly in multidrug-resistant Staphylococcus aureus

枯草芽孢杆菌衍生的肽会破坏多重耐药金黄色葡萄球菌的群体感应和生物膜组装

Leistikow, Kyle R; May, Daniel S; Suh, Won Se; Vargas Asensio, Gabriel; Schaenzer, Adam J; Currie, Cameron R; Hristova, Krassimira R

Angucyclinones rescue PhLOPSA antibiotic activity by inhibiting Cfr-dependent antibiotic resistance

Angucyclinones 通过抑制 Cfr 依赖性抗生素耐药性来挽救 PhLOPSA 抗生素活性

Adam J Schaenzer, Annia Rodriguez Hernandez, Kaitlyn Tsai, Christian Hobson, Danica Galonić Fujimori, Gerard D Wright

Current Insights into the Steroidal Module of the Athlete Biological Passport

运动员生物护照中类固醇模块的最新见解

Piper, Thomas; Geyer, Hans; Haenelt, Nadine; Huelsemann, Frank; Schaenzer, Wilhelm; Thevis, Mario

GW779439X and Its Pyrazolopyridazine Derivatives Inhibit the Serine/Threonine Kinase Stk1 and Act As Antibiotic Adjuvants against β-Lactam-Resistant Staphylococcus aureus

GW779439X 及其吡唑并哒嗪衍生物抑制丝氨酸/苏氨酸激酶 Stk1 并作为抗 β-内酰胺耐药金黄色葡萄球菌的抗生素佐剂

Adam J Schaenzer, Nathan Wlodarchak, David H Drewry, William J Zuercher, Warren E Rose, Carla A Ferrer, John-Demian Sauer, Rob Striker

In Silico Screen and Structural Analysis Identifies Bacterial Kinase Inhibitors which Act with β-Lactams To Inhibit Mycobacterial Growth

通过计算机筛选和结构分析鉴定出与 β-内酰胺一起抑制分枝杆菌生长的细菌激酶抑制剂

Nathan Wlodarchak, Nathan Teachout, Jeffrey Beczkiewicz, Rebecca Procknow, Adam J Schaenzer, Kenneth Satyshur, Martin Pavelka, William Zuercher, David Drewry, John-Demian Sauer, Rob Striker

A screen for kinase inhibitors identifies antimicrobial imidazopyridine aminofurazans as specific inhibitors of the Listeria monocytogenes PASTA kinase PrkA

激酶抑制剂筛选鉴定出抗菌咪唑并吡啶氨基呋喃并物是单核细胞增生李斯特菌 PASTA 激酶 PrkA 的特异性抑制剂

Adam J Schaenzer, Nathan Wlodarchak, David H Drewry, William J Zuercher, Warren E Rose, Rob Striker, John-Demian Sauer

The Listeria monocytogenes PASTA Kinase PrkA and Its Substrate YvcK Are Required for Cell Wall Homeostasis, Metabolism, and Virulence

单核细胞增生李斯特菌 PASTA 激酶 PrkA 及其底物 YvcK 是细胞壁稳态、代谢和毒力所必需的

Pensinger, Daniel A; Boldon, Kyle M; Chen, Grischa Y; Vincent, William J B; Sherman, Kyle; Xiong, Meng; Schaenzer, Adam J; Forster, Emily R; Coers, Jörn; Striker, Rob; Sauer, John-Demian

Selective pharmacologic inhibition of a PASTA kinase increases Listeria monocytogenes susceptibility to β-lactam antibiotics

选择性药物抑制 PASTA 激酶可增加单核细胞增生李斯特菌对 β-内酰胺类抗生素的敏感性

Daniel A Pensinger, Matthew T Aliota, Adam J Schaenzer, Kyle M Boldon, Israr-ul H Ansari, William J B Vincent, Benjamin Knight, Michelle L Reniere, Rob Striker, John-Demian Sauer