日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting HER2-Positive HCC1954 Breast Cancer Cells by Novel Thiazole-Dihydrobenzisoxazoles: In-Depth Design, Synthesis and Initial In Vitro Study

利用新型噻唑-二氢苯并异噁唑靶向HER2阳性HCC1954乳腺癌细胞:深入设计、合成及初步体外研究

Piven, Yuri A; Sorokin, Danila V; Varabyeva, Nastassia A; Mikhaylova, Alexandra L; Bogdanov, Fedor B; Shafranovskaya, Elena V; Puzanau, Raman M; Lakhvich, Fedor A; Scherbakov, Alexander M

Secosteroid-2-Pyrazoline Hybrids: Design, Synthesis, Biological Evaluation and Development of Therapeutic Combinations Against ERα-Positive Breast Cancer Cells

甾体-2-吡唑啉杂合物:设计、合成、生物学评价及针对ERα阳性乳腺癌细胞的治疗组合开发

Ilovaisky, Alexey I; Scherbakov, Alexander M; Bogdanov, Fedor B; Miciurov, Dumitru; Chernoburova, Elena I; Merkulova, Valentina M; Bozhenko, Eugene I; Dmitrenok, Andrey S; Salnikova, Diana I; Sorokin, Danila V; Khamidullina, Alvina I; Krasil'nikov, Mikhail A; Zavarzin, Igor V; Terent'ev, Alexander O

Novel N-(4,5,6,7-tetrahydrobenzisoxazol-4-yl)amides as HSP90 inhibitors: design, synthesis and biological evaluation.

新型 N-(4,5,6,7-四氢苯并异噁唑-4-基)酰胺作为 HSP90 抑制剂:设计、合成和生物学评价

Varabyeva Nastassia A, Scherbakov Alexander M, Salnikova Diana I, Sorokin Danila V, Khamidullina Alvina I, Mikhaylova Alexandra L, Paulovich Dzmitry I, Lakhvich Fedor A, Piven Yuri A

Breast cancer cell resistance to hormonal and targeted therapeutics is correlated with the inactivation of the NR6A1 axis

乳腺癌细胞对激素和靶向治疗的耐药性与NR6A1轴的失活相关。

Andreeva, Olga E; Sorokin, Danila V; Vinokurova, Svetlana V; Kopnin, Pavel B; Elkina, Nadezhda V; Katargin, Alexey N; Faskhutdinov, Radik S; Salnikova, Diana I; Scherbakov, Alexander M; Krasil'nikov, Mikhail A

Synthesis and evaluation of sulfonamide derivatives of quinoxaline 1,4-dioxides as carbonic anhydrase inhibitors

喹喔啉1,4-二氧化物磺酰胺衍生物的合成及作为碳酸酐酶抑制剂的评价

Buravchenko, Galina I; Scherbakov, Alexander M; Krymov, Stepan K; Salnikova, Diana I; Zatonsky, George V; Schols, Dominique; Vullo, Daniela; Supuran, Claudiu T; Shchekotikhin, Andrey E

Synthesis and Biological Evaluation of Chalconesulfonamides: En Route to Proapoptotic Agents with Antiestrogenic Potency

查尔酮磺酰胺的合成及生物学评价:通往具有抗雌激素活性的促凋亡剂之路

Krymov, Stepan K; Salnikova, Diana I; Dezhenkova, Lyubov G; Bogdanov, Fedor B; Korlyukov, Alexander A; Scherbakov, Alexander M; Shchekotikhin, Andrey E

Honokiol inhibits the growth of hormone-resistant breast cancer cells: its promising effect in combination with metformin

厚朴酚抑制激素抵抗性乳腺癌细胞的生长:其与二甲双胍联合使用具有良好的效果

Mikhaevich, Ekaterina I; Sorokin, Danila V; Scherbakov, Alexander M

Design, Synthesis and In Vitro Investigation of Cabozantinib-Based PROTACs to Target c-Met Kinase

基于卡博替尼的PROTAC靶向c-Met激酶的设计、合成及体外研究

Sachkova, Anastasia A; Andreeva, Daria V; Tikhomirov, Alexander S; Scherbakov, Alexander M; Salnikova, Diana I; Sorokin, Danila V; Bogdanov, Fedor B; Rysina, Yulia D; Shchekotikhin, Andrey E; Shchegravina, Ekaterina S; Fedorov, Alexey Yu

Novel d-Annulated Pentacyclic Steroids: Regioselective Synthesis and Biological Evaluation in Breast Cancer Cells

新型d-稠合五环甾体:区域选择性合成及在乳腺癌细胞中的生物学评价

Vorontsova, Svetlana K; Yadykov, Anton V; Scherbakov, Alexander M; Minyaev, Mikhail E; Zavarzin, Igor V; Mikhaevich, Ekaterina I; Volkova, Yulia A; Shirinian, Valerii Z

Exosome-Mediated Transfer of Cancer Cell Resistance to Antiestrogen Drugs

外泌体介导的癌细胞抗雌激素药物耐药性转移

Semina, Svetlana E; Scherbakov, Alexander M; Vnukova, Anna A; Bagrov, Dmitry V; Evtushenko, Evgeniy G; Safronova, Vera M; Golovina, Daria A; Lyubchenko, Ludmila N; Gudkova, Margarita V; Krasil'nikov, Mikhail A