日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An all-in-one pipeline for the in vitro discovery and in vivo testing of Plasmodium falciparum malaria transmission blocking drugs.

用于体外发现和体内测试恶性疟原虫疟疾传播阻断药物的一体化流程

Brancucci Nicolas M B, Gumpp Christin, van Gemert Geert-Jan, Yu Xiao, Passecker Armin, Nardella Flore, Thommen Basil T, Chambon Marc, Turcatti Gerardo, Halby Ludovic, Blasco Benjamin, Duffey Maëlle, Arimondo Paola B, Bousema Teun, Scherf Artur, Leroy Didier, Kooij Taco W A, Rottmann Matthias, Voss Till S

Ectopic overexpression of Plasmodium falciparum DNA-/RNA-binding Alba proteins misregulates virulence gene homeostasis during asexual blood development

恶性疟原虫DNA/RNA结合蛋白Alba的异位过表达会在无性血液发育过程中扰乱毒力基因的稳态。

Acharya, Dimple; Bavikatte, Anitha Nagaraj; Ashok, Vishnu Vinayak; Hegde, Shubhada R; Macpherson, Cameron Ross; Scherf, Artur; Vembar, Shruthi Sridhar

Plasmodium-encoded murine IL-6 impairs liver stage infection and elicits long-lasting sterilizing immunity

疟原虫编码的小鼠IL-6可抑制肝期感染并诱导持久的清除性免疫。

Belhimeur, Selma; Briquet, Sylvie; Peronet, Roger; Pham, Jennifer; Commere, Pierre-Henri; Formaglio, Pauline; Amino, Rogerio; Scherf, Artur; Silvie, Olivier; Mecheri, Salaheddine

Humanized mice for investigating sustained Plasmodium vivax blood-stage infections and transmission

利用人源化小鼠研究间日疟原虫持续性血液期感染和传播

Luiza-Batista, Camilla; Thiberge, Sabine; Serra-Hassoun, Malika; Nardella, Flore; Claës, Aurélie; Nicolete, Vanessa C; Commère, Pierre-Henri; Mancio-Silva, Liliana; Ferreira, Marcelo U; Scherf, Artur; Garcia, Sylvie

DNA Methylation Bisubstrate Inhibitors Are Fast-Acting Drugs Active against Artemisinin-Resistant Plasmodium falciparum Parasites

DNA甲基化双底物抑制剂是速效药物,可有效对抗青蒿素耐药的恶性疟原虫。

Nardella, Flore; Halby, Ludovic; Hammam, Elie; Erdmann, Diane; Cadet-Daniel, Véronique; Peronet, Roger; Ménard, Didier; Witkowski, Benoit; Mecheri, Salah; Scherf, Artur; Arimondo, Paola B

Development of a Photo-Cross-Linkable Diaminoquinazoline Inhibitor for Target Identification in Plasmodium falciparum

开发一种光交联二氨基喹唑啉抑制剂用于恶性疟原虫靶标识别

Lubin, Alexandra S; Rueda-Zubiaurre, Ainoa; Matthews, Holly; Baumann, Hella; Fisher, Fabio R; Morales-Sanfrutos, Julia; Hadavizadeh, Kate S; Nardella, Flore; Tate, Edward W; Baum, Jake; Scherf, Artur; Fuchter, Matthew J

Modifications at K31 on the lateral surface of histone H4 contribute to genome structure and expression in apicomplexan parasites.

组蛋白 H4 侧面 K31 位点的修饰有助于顶复门寄生虫的基因组结构和表达

Sindikubwabo Fabien, Ding Shuai, Hussain Tahir, Ortet Philippe, Barakat Mohamed, Baumgarten Sebastian, Cannella Dominique, Palencia Andrés, Bougdour Alexandre, Belmudes Lucid, Couté Yohann, Tardieux Isabelle, Botté Cyrille Y, Scherf Artur, Hakimi Mohamed-Ali

Trans-acting GC-rich non-coding RNA at var expression site modulates gene counting in malaria parasite

反式作用的富含GC的非编码RNA在var表达位点调节疟原虫的基因计数

Guizetti, Julien; Barcons-Simon, Anna; Scherf, Artur

Translational regulation in blood stages of the malaria parasite Plasmodium spp.: systems-wide studies pave the way

疟原虫血液期翻译调控:系统性研究为其铺平道路

Vembar, Shruthi Sridhar; Droll, Dorothea; Scherf, Artur

Original 2-(3-Alkoxy-1H-pyrazol-1-yl)azines Inhibitors of Human Dihydroorotate Dehydrogenase (DHODH)

原始的 2-(3-烷氧基-1H-吡唑-1-基)嗪类人二氢乳清酸脱氢酶 (DHODH) 抑制剂

Lucas-Hourani, Marianne; Munier-Lehmann, Hélène; El Mazouni, Farah; Malmquist, Nicholas A; Harpon, Jane; Coutant, Eloi P; Guillou, Sandrine; Helynck, Olivier; Noel, Anne; Scherf, Artur; Phillips, Margaret A; Tangy, Frédéric; Vidalain, Pierre-Olivier; Janin, Yves L